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6-(5-methylfuran-2-yl)-3,4-dihydroquinazolin-4-one
1-(3-chlorophenyl)-4-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperazin-2-one
methyl 1-[3-(2-methyl-1H-indol-1-yl)propanoyl]azetidine-3-carboxylate
3-(4-hydroxyphenyl)-N-methyl-N-(quinolin-5-ylmethyl)benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-acetamido-3-hydroxypropanamide
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(1H-pyrazol-1-yl)phenyl]urea
2-[3-(methoxymethyl)phenyl]-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-cyclobutyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 5-(cyclopropylmethyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[(1-methanesulfonylpiperidin-4-yl)amino]-N,N-bis(prop-2-en-1-yl)acetamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylpyrazine-2-carboxamide
4-methyl-2-[1-(1-methyl-1H-indole-6-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
(3S,4S)-4-propyl-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}methyl)pyrrolidin-3-ol
2-{2-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[4-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)phenyl]acetamide
6-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-cyclopropyl-6-(2-fluorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]piperidine
N-{2-[bis(propan-2-yl)amino]ethyl}-6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 2-{4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholin-3-yl}acetate
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}pyrimidin-2-amine
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-5-hydroxypyrazine-2-carboxamide
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(6-methoxypyridin-3-yl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
4-(pyrimidin-2-yl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
3-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-N-(propan-2-yl)propanamide
(2S,3R)-2-amino-1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-methoxybutan-1-one
4-(2-fluorophenyl)-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
5-methoxy-2-(3-methyl-1-phenyl-1H-1,2,4-triazol-5-yl)phenol
N,N-dimethyl-3-[3-(piperidine-1-carbonyl)pyridin-2-yl]aniline
N4-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidine-4,6-diamine
methyl 2-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
1-(2-fluorophenyl)-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazine
N-(furan-3-ylmethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-(1-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)isoquinoline
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-3-yl}propanamide
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-5-methoxy-3-methyl-1H-indole
1-cyclopentyl-4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrrolidin-2-one
5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-1-[(2,4-difluorophenyl)methyl]azepan-2-one
1-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
15-methyl-13-oxo-N-[3-(pyridin-4-yl)propyl]-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-(piperidin-3-ylmethyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}propanamide
4-{[5-(oxan-2-yl)furan-2-yl]methyl}-1-phenylpiperazin-2-one