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3-(6-cyanopyridin-3-yl)-1-[(1-hydroxycyclohexyl)methyl]urea
8-{[2-(furan-2-yl)phenyl]methyl}-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentanecarbonyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
(2E)-N-{1-[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]propan-2-yl}-3-phenylprop-2-enamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
2-(methylsulfanyl)-N-(pyridin-2-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-(1-{1-[(2-chloro-5-fluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}propyl)-N-methylacetamide
6-(aminomethyl)-2-[3-({[(3-chlorophenyl)methyl](cyclopropyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3,5-dimethyl-N-[2-(methylsulfanyl)ethyl]-1-benzofuran-2-carboxamide
[4-({[(5-fluoro-3-methyl-1H-indol-2-yl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
methyl 2-({6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)benzoate
3-(1H-1,2,4-triazol-1-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}adamantane-1-carboxamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1'-cyclohexyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1-methyl-1H-imidazol-2-yl)({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl})methanol
N-(1-methoxypropan-2-yl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl)[(3-methylpyridin-4-yl)methyl]amine
1-cyclopropyl-3-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-[(3-hydroxyphenyl)methyl]urea
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-methylfuran-3-carboxamide
1-(1,3-benzothiazol-5-yl)-3-methyl-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
3-(2,1,3-benzothiadiazol-5-ylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
N-ethyl-4-phenyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]butanamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
3-butyl-4-[(3-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]-2,1,3-benzoxadiazole
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
ethyl 2-{2-[(2-benzamido-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl)formamido]ethyl}-1,3-thiazole-4-carboxylate
5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridine-2-carbonitrile
(3R,4S)-4-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
8-{2-[(dimethylamino)methyl]benzoyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[2-(thiophen-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(5-chloropyridin-2-yl)-4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperazine
N-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
2-(4-{[2-hydroxy-2-(pyridin-2-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
N-[2-(methylsulfanyl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
N-({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}methyl)acetamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(2S,4R)-4-acetamido-N,N-diethyl-1-[4-(propan-2-yl)benzoyl]pyrrolidine-2-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
3-{[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}-2,2-dimethylpropan-1-ol
12-[(3S)-3-ethylmorpholine-4-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
3-(4-fluorophenoxymethyl)-N-(2-methoxypyridin-3-yl)piperidine-1-carboxamide