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(1R,5S,6R)-3-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
9-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}amine
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-4-(trifluoromethyl)benzamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-({1-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]cyclopropyl}methyl)-1H-pyrazole
methyl(quinoxalin-2-ylmethyl)[(2,3,4-trifluorophenyl)methyl]amine
N-(1-benzothiophen-2-ylmethyl)-N-methyloxolane-3-carboxamide
2-methyl-N4-[4-(pyrrolidin-1-yl)butyl]pyrimidine-4,6-diamine
4-({2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxamide
1-(3-methoxyphenyl)-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperazin-2-one
2-benzyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,1-dimethyl-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyridine-3-carboxamide
(3aR,6aR)-2-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-butyl-N-methyl-3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-cyclohexyl-4-(2,5-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]phenyl}propanoic acid
dimethyl[3-(2-{1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
6-[3-(2-methylphenoxymethyl)piperidin-1-yl]pyrimidine-2,4-diamine
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
N,2-dimethyl-N-(1-methylpyrrolidin-3-yl)-4-phenylpyridine-3-carboxamide
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-propyl-N-(thiophen-3-ylmethyl)acetamide
6-(methoxymethyl)-N,1-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{4-[(4-methylphenyl)methyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}-1,4-diazepane-1-carbaldehyde
2-amino-3-ethyl-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[2-({4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}methyl)morpholin-4-yl]ethan-1-one
N-methyl-2-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxaspiro[4.4]nonane-4-carboxamide
1-phenyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepane
1-ethyl-3-(2-methylpropyl)-N-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
1-(2,2-dimethylpropyl)-3-[(4-ethylpiperazin-1-yl)methyl]-3-hydroxypiperidin-2-one
5-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-{1-[3-(pyridin-3-yl)propyl]piperidin-3-yl}benzoic acid
N-[2-(N-methylmethanesulfonamido)ethyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
8-(2-fluorobenzenesulfonyl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
[(3R,4R)-1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-4-(azepan-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(3,4-difluorophenyl)-6-[4-(morpholin-4-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
2-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4R)-4-amino-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidine-2-carboxamide
3-fluoro-N-[3-(1H-imidazol-1-yl)propyl]-7-methylimidazo[1,2-a]pyridine-2-carboxamide
7-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-2,7-diazaspiro[4.5]decane
2,4-dimethoxy-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-indole-2-carboxamide
benzyl (7S,9aR)-7-[(benzyloxy)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-methyl-1'-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
{3-[(2,4-difluorophenyl)methyl]-1-[4-(piperidin-1-yl)benzoyl]piperidin-3-yl}methanol