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(1R,7S)-3-(2,2-dimethylpropyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-N-phenylpiperidin-3-amine
N-ethyl-1-methyl-3-(2-methylpropyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(1R,2S,9R)-11-(2-methyl-5-propylpyrimidin-4-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(2-hydroxyethyl)-6-[2-(1-propylpiperidin-4-yl)acetyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
2-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)propanamide
{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}[(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
2-(4-ethylpiperazin-1-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
8-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
4-(4-chlorophenoxy)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
7-(3-chlorophenyl)-9-hydroxy-N,N-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-1,4-diazepan-5-one
(2R,3S)-2-amino-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-hydroxybutan-1-one
N-[(1-{[4-(methylsulfamoyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
1-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
4-[3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)propanoyl]-3,3-dimethylpiperazin-2-one
2-benzyl-8-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
3-(1-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyridine
2-(furan-2-yl)-2-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(1R,5S)-8-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
7-(cyclopropylmethyl)-2-(2-methoxypyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-3-cyclopentyl-1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(cyclopentylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3-{[(4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
1-[2-(4-methoxyphenyl)ethyl]-5-(2-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(quinoline-3-carbonyl)pyrrolidine-2-carboxamide
N-(9H-fluoren-9-yl)imidazo[1,2-a]pyrimidine-2-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-amine
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
N4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N4,N6,N6-trimethylpyrimidine-4,6-diamine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(trifluoromethyl)benzamide
3-(3-methylphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methylacetamide
N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-6-methylpyridine-3-carbonitrile
2-methoxy-1-{1'-[2-(propylsulfanyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(2-oxopyrrolidin-1-yl)benzamide
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-phenylbutan-1-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
6-cyano-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-3-carboxamide
9-(4,6-dimethylpyrimidin-2-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-5-cyclopentyl-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide