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4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-7-methylquinoline
1-(4-{[4-(4-hydroxyphenyl)butan-2-yl]amino}piperidin-1-yl)-2-methylpropan-1-one
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
3-benzyl-4-(prop-2-en-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-1H-imidazole-4-carboxylic acid
ethyl 3-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-methylpentanoate
4-{[1-(1,3-thiazol-2-yl)piperidin-3-yl]methyl}benzoic acid
(1R,5R)-3-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N,N-bis(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl 5-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-5-oxopentanoate
1-{2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-1,2-dihydroquinoxalin-2-one
4-[1-(1-cyclopropylethyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-(3-fluorophenyl)-1H-pyrazole
6-(4-oxo-4-phenylbutanoyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
[(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-(furan-2-ylmethyl)-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]piperidine
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-cyclopentyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(5-chlorothiophen-2-yl)methyl]-3-(pyridin-4-yl)propanamide
2-(4-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
N-(2-methoxy-6-methylphenyl)-3-[(3-methylpiperidin-1-yl)methyl]benzamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
[(3R,4R)-1-[4-(difluoromethoxy)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-methyl-2-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-2-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidine
N-[2-(3,5-dimethoxyphenyl)ethyl]-1-methylpiperidine-2-carboxamide
1-(4-chloro-2-ethylphenyl)-3-methyl-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
3-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methoxy]-2-ethyl-6-methylpyridine
4-hydroxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
9-(4-methylnaphthalene-1-carbonyl)-3,9-diazaspiro[5.6]dodecane
dimethyl(2-{2-[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]-1H-imidazol-1-yl}ethyl)amine
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-(adamantan-2-yl)-6-{[butyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperazin-2-one
2-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
3-cyclopropyl-4-[3-ethoxy-4-methoxy-5-(prop-2-en-1-yl)phenyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-1,3-benzodiazole-5-carboxamide
methyl 3-methyl-4-({[2-methyl-1-(pyridin-3-yl)propyl]carbamoyl}amino)benzoate
2-[2-methyl-3-({[(1S)-1-phenylpropyl]amino}methyl)-1H-indol-1-yl]acetamide
(2S,4R)-4-amino-1-(2,6-dimethoxypyrimidine-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
2-(3-acetyl-1H-indol-1-yl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(2-oxoazepan-1-yl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(2-ethoxyphenyl)-3-hydroxypiperidine-1-carboxamide
(3S,4S)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1,3-dimethyl-6-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(furan-2-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2-methyl-6-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid