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N-[(3S,4R)-1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-3,4-dihydroquinazolin-4-one
ethyl 2-(1-{1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-amido}cyclohexyl)acetate
4-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-6-(1H-pyrazol-1-yl)pyrimidine
N-[1-(thian-4-yl)piperidin-4-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(benzylamino)-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
N-(2-methoxyethyl)-2-(1H-pyrazol-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(2-methoxyethyl)-2-(methylamino)-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-cyclopropyl-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(pyridin-4-ylmethyl)benzamide
5-chloro-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyridine-2-carboxamide
5-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-(2-chlorophenyl)-N-[3-(dimethylamino)propyl]-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(2-hydroxyethyl)-3-(pyridin-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-(4-fluorophenoxymethyl)-N-(4-hydroxybutan-2-yl)-N-methyl-1,3-oxazole-4-carboxamide
3-{1-[1-(cyclohexylcarbamoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propanoic acid
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
7-[cyclohexyl(methoxy)methyl]-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(cyclohexylmethyl)acetamide
2-ethyl-8-(4-oxo-4-phenylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-5,6-dihydro-1,4-dioxine-2-carboxamide
2-(2H-indazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propylfuran-2-carboxamide
1-[(3-methylphenyl)methyl]-4-[3-(piperidin-3-yl)benzoyl]piperazin-2-one
1-{4-[(2,6-difluoro-3-methylphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
8-[(5-hydroxy-2-methoxyphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]piperidin-3-yl}benzoic acid
3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
2-[(2-phenylethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
4-chloro-N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,1-dimethyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-(2-fluorophenoxymethyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
3-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)benzoic acid
N-methyl-5-phenyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]prop-2-en-1-one
1-[2-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-methyl-2-oxo-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
3-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
2,5-dimethyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(2-methoxyethyl)piperazine