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6,7-dimethoxy-2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
1-(4-{[2-(3-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}piperazin-1-yl)ethan-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetyl}pyrrolidine-2-carboxamide
3-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
methyl 3-benzamido-5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3,5-difluoro-N-[2-(1,3-thiazol-2-yl)ethyl]pyridine-2-carboxamide
6-[5-(methanesulfonylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
(1R,2R,4R)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-(hydroxymethyl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azepan-4-ol
methyl 4-({[2-(dimethylamino)pyridin-3-yl]methyl}carbamoyl)benzoate
3-(4-fluorophenyl)-4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-pyrazole
5-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-4-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
5-(2,6-dimethoxyphenyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2,4-triazin-3-amine
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(cyclohexylmethyl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-butyl-4-[2-(3-hydroxyazetidin-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-oxopiperidin-1-yl)propanamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
1-(2-benzylmorpholin-4-yl)-2-cyclopropylethan-1-one
5-[3-(methoxymethyl)piperidine-1-carbonyl]-2-[4-(propan-2-yl)piperidin-1-yl]pyridine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(3-phenylpropyl)piperidine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-phenyl-1H-1,2,3-triazole
N-methyl-N'-(4-methylphenyl)-N-[1-(1,3-thiazol-2-yl)ethyl]propanediamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(quinoxalin-2-yl)piperidin-3-ol
4-tert-butyl-6-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
(3S,4S)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-{3-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}ethan-1-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
8-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-cyclopentyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}pyrimidine
4-benzoyl-N-(3-benzyl-1H-1,2,4-triazol-5-yl)piperazine-1-carboxamide
1-[4-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-ethyl-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-hydroxy-5-{[2-(2-phenylethyl)morpholin-4-yl]methyl}benzoic acid
8-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}quinoline
methyl 4-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]butanoate
2-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyridine-3-carbonitrile
(3aR,6aR)-2-methanesulfonyl-5-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(methoxymethyl)-N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidin-4-amine
N-ethyl-2-(4-fluorophenoxymethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
6-[(2,3-difluoro-4-methylphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-[3-oxo-9-(pyridine-3-sulfonyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid