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1-(5-chloro-2-methylphenyl)-3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
methyl 1-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-2-carboxylate
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)pent-4-enamide
4-{4-[(furan-2-ylmethyl)amino]piperidin-1-yl}-N-(1-phenylethyl)benzamide
(2S)-2-[(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)formamido]propanamide
(1R,5R)-6-(cyclopropylmethyl)-3-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-methoxypropanamide
N-methyl-2-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-N-(propan-2-yl)acetamide
ethyl 4-(3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-6,7-dimethoxyquinolin-2-yl)piperazine-1-carboxylate
5-cyclopropanecarbonyl-1'-(5-methyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(1-hydroxy-2-{4-[2-(5-methylfuran-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)phenol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(dicyclopropylmethyl)acetamide
(1S,5R)-6-benzyl-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
1-methyl-3-(propan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5,6-dimethylpyridine-3-carbonitrile
1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]piperidine-2-carboxylic acid
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[4-(4-fluorophenyl)benzoyl]-1,4-diazepan-5-one
4-benzyl-3-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-2-[(3,5-dimethyl-1H-indol-2-yl)formamido]-4-(methylsulfanyl)butanoic acid
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-cyclopropyl-3-(5-{imidazo[1,2-a]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
methyl 5-{[(4-fluorophenyl)carbamoyl]carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-{[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
3-[(5-ethylpyridin-2-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
5-ethyl-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-2-(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)-1H-1,3-benzodiazole
N-cyclopropyl-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-4-carboxamide
N-{4-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
5-(1-{[4-(hydroxymethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-2-methoxybenzoic acid
2,6-dimethoxy-N-(1-methyl-5-oxopyrrolidin-3-yl)pyrimidine-4-carboxamide
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]urea
(3S,4R)-1-(cyclopropanesulfonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-[(3S,4R)-1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-(4-methoxyphenyl)-4-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
1-methyl-3-(propan-2-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-methyl-8-(2-phenoxybenzoyl)-2,8-diazaspiro[4.5]decan-3-one
[2-(4-fluorophenyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-hydroxypropan-2-yl)acetamide
2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
N-(furan-2-ylmethyl)-2-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]acetamide
2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyridine-4-carboxamide
(1S,5R)-1,3,3-trimethyl-6-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-6-azabicyclo[3.2.1]octane
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(4-methyl-1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1S,6R)-9-{[5-(2-chlorophenyl)furan-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
ethyl 2-[4-(1H-pyrazol-5-yl)phenyl]pyridine-3-carboxylate
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
4-[(8-methoxyquinolin-2-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide