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(2S)-2-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylethan-1-ol
2-(2-methylphenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-[(3R,4S)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
6-[(diethylamino)methyl]-N-(1H-indol-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(1-{5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazol-3-yl}-N-methylformamido)-N-methylacetamide
N-cyclopropyl-3-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}propanamide
1-(4-{[(1S,2S)-2-hydroxycyclohexyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(3R,4S)-1-(3-chloropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-amine
1-(cyclohexylmethyl)-N-(2,2-diphenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
2-methoxy-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-ethyl-1,3,4-oxadiazol-2-amine
ethyl 3-benzyl-1-(1,4-dithiepan-6-yl)piperidine-3-carboxylate
2-methyl-6-(2-phenylethyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1'-[(8-methoxy-2H-chromen-3-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
1-cyclohexyl-4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
2-[2-(2-fluorophenyl)ethyl]-4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-methoxyphenyl)-1,2,4-oxadiazole
N-[(3-methoxyphenyl)methyl]-3-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-yl]propanamide
6-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N,N-dimethylpyrazine-2-carboxamide
1-(3-methoxyphenyl)-5-methyl-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-2-one
4-cyclohexyl-N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-1,4-diazepane-1-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-{2-[2-(4-methylpentyl)morpholin-4-yl]-2-oxoethyl}pyrrolidin-2-one
ethyl 2-[4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)morpholin-3-yl]acetate
N'-(2-ethoxyphenyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]propanediamide
N-[2-(2,6-dichlorophenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[3-(1H-indol-1-yl)propyl]-5-methylpyrazine-2-carboxamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(3S,4R)-1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4-propylpyrrolidin-3-yl]acetamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-methyl-N-{3-[methyl(phenyl)amino]propyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(4-hydroxyphenyl)propan-1-one
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 6-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-3-carboxylate
N-(quinolin-6-yl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
3-(4-hydroxyphenyl)-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]propanamide
3-methoxy-N-[(2-methoxyphenyl)methyl]-N-propylpropanamide
N-ethyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N4-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidine-3-carboxamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxan-2-ylmethyl)pyridin-2-amine
6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(2-fluorophenyl)ethyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
1-{2-[3-(2-methylphenoxy)azetidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
N-(2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)acetamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-3-yl)acetamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidine
(2S,4R)-4-amino-N-ethyl-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide