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N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-1-methylpiperidine-2-carboxamide
1-(cyclobutylmethyl)-3-{[(cyclohexylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
3-[4-(1-ethyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(2-ethylphenyl)propanamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)methylamine
1-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}benzoyl)-4-methyl-1,2,3,6-tetrahydropyridine
(4aR,8aR)-2-[4-(dimethylamino)benzoyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-[2-(pyridin-3-yl)ethyl]propanamide
1-[2-methyl-2-(pyrrolidin-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N'-(4-methylphenyl)-N-[2-(pyridin-3-yloxy)propyl]propanediamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)urea
2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]pyridine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(1H-pyrazol-4-yl)pyridine-3-carboxamide
(3R,4R)-1-(azepane-1-sulfonyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
N-(2-fluoroethyl)-3-[methyl(1-methylpyrrolidin-3-yl)sulfamoyl]benzamide
1-ethyl-N-[(4-phenyloxan-4-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
5-cyclopropanecarbonyl-1'-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 6-{6-oxo-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}pyridine-2-carboxylate
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-benzofuran-3-carboxamide
N-(3-cyano-4-ethoxyphenyl)-4-(pyrimidin-4-yl)piperidine-1-carboxamide
5-[3-(4-ethylphenyl)propyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(2,3-dihydro-1-benzofuran-5-yl)-2-propyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-[(dimethylamino)methyl]-4-[1-(quinolin-3-yl)-1H-imidazol-2-yl]phenol
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
4-(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-2-methylpyrimidine
1-(2-methyloxane-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-4-carboxamide
9-[(4-methoxy-3-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
5-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]pyridine-2-carbonitrile
4-(4-carbamoylphenyl)-3-methylbenzoic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane
1-[(2-hydroxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-[3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
9-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}pyrazine
1-[4-(morpholin-4-yl)-3-(oxan-2-ylmethyl)phenyl]ethan-1-one
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
1-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
1-[(4-fluorophenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,4-diazepane
N-cyclopentyl-N'-(quinolin-3-ylmethyl)butanediamide
2-(1H-1,2,4-triazol-3-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}benzamide
4-[5-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
N-[2-(ethylsulfanyl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-cyclopentyl-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
(2S)-2-{[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazol-3-yl]formamido}propanamide
2-benzyl-8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one