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ethyl 3-[(3-chlorophenyl)methyl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine-3-carboxylate
N,1-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
N-{2-[cyclopentyl(methyl)amino]ethyl}-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
(2S)-1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3S,5S)-1-[(2E)-3-phenylprop-2-en-1-yl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(4,6-dimethylpyridin-3-yl)methyl]propanamide
1-methyl-8-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(3aR,6aR)-2-cyclopentyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1S,5R)-6-benzyl-3-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-[4-(adamantan-2-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-(2-ethoxyphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
2-{4-[2-(pyridin-2-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-methyl-1-{2-oxo-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}-1,4-dihydroquinolin-4-one
1-cyclohexyl-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-(3-methyl-1,2-oxazol-5-yl)-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
methyl 4-(2-amino-6-tert-butyl-3-cyanopyridin-4-yl)-1H-pyrazole-3-carboxylate
4,6-dimethyl-13-[2-(propylamino)pyrimidin-5-yl]-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
[4-fluoro-3-(isoquinolin-5-yl)phenyl]methanamine
6-[(3,5-dimethoxyphenyl)methoxy]-4-(oxan-4-yl)-1-(propan-2-yl)-1,4-diazepan-2-one
2-{4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenoxy}ethan-1-ol
5-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-[(2S)-pyrrolidin-2-ylmethyl]-3-[(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
2-{2-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
9-(cyclopropylmethyl)-4-[(3-fluoro-2-methylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-hydroxy-N-[3-(pyridin-3-yl)propyl]pyridine-2-carboxamide
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-4-methoxyphenol
1-benzyl-8-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-9-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxy-1-oxopropan-2-yl}acetamide
4,6-dimethyl-1-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(2R,6R)-4-acetyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{4-oxo-4-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butyl}piperidin-2-one
2-(adamantan-1-ylsulfanyl)-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(2,2-dimethyl-4-phenyloxan-4-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[3-(1H-1,2,4-triazol-1-yl)propyl]amine
2,6-dimethyl-3-[3-(1H-pyrazol-3-yl)phenyl]pyridine
1-{6-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyridin-2-yl}ethan-1-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[(3-hydroxyazetidin-1-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
(3S,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
1-methyl-1-({3-[2-(methylsulfanyl)ethyl]-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)urea
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2-ethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide