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N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-sulfamoylbutanamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-cyclopentyl-N3-ethyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
(3S)-4-[(5-acetylthiophen-3-yl)methyl]-3-benzylpiperazin-2-one
1-cyclopropyl-4-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)pyrrolidin-2-one
N-(1-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-4-yl)methanesulfonamide
5-[6-chloro-4-(1,4-oxazepane-4-carbonyl)quinolin-2-yl]pyrimidin-2-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(1H-indol-3-yl)-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(3-chlorophenyl)-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
4-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
5-acetyl-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopentylacetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxylate
1-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-oxopiperidine-3-carboxamide
1-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
(1R,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxyethyl 4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperidin-4-ol
2-benzyl-8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amine
3-ethyl-1-{2-methoxy-4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}urea
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-2-carboxamide
4-{4-[(6-methoxypyrimidin-4-yl)amino]piperidin-1-yl}-1λ6-thiane-1,1-dione
(3R,4R)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(morpholin-4-yl)piperidin-3-ol
(2S)-1-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)propan-2-ol
N-(2,4-dimethylphenyl)-2-({3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}amino)acetamide
6-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(prop-2-en-1-yl)acetamide
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[(1R)-1-(4-chlorophenyl)ethyl]urea
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-N'-(3-chloro-4-fluorophenyl)propanediamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-(methoxymethyl)furan-2-carboxamide
N-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}methanesulfonamide
N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]acetamide
(4aS,8aR)-N-cyclopentyl-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
4-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-2-yl}methyl)morpholine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(dimethylamino)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methylpropanamide
N4-[3-(furan-2-yl)phenyl]-N1-(furan-2-ylmethyl)piperidine-1,4-dicarboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propan-1-one