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[5-fluoro-7-(quinolin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-1H-1,2,3-benzotriazole-5-carboxamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(2-phenylethyl)piperidine
1-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-3-ethyl-3-(oxolan-2-ylmethyl)urea
N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methyl-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thieno[2,3-d]pyrimidin-4-amine
methyl 6-[propyl(pyridin-3-ylmethyl)carbamoyl]pyridine-3-carboxylate
{1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-[2-(2-fluorophenyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-cyclobutanecarbonyl-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(3-methoxyphenyl)methyl]-4-[(trimethylpyrazin-2-yl)methyl]morpholine
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-4-oxobutanamide
N-(2H-1,3-benzodioxol-5-yl)piperidin-3-amine
3-[4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenyl]prop-2-yn-1-ol
2-{5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
3-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-[4-(propylsulfamoyl)phenyl]urea
1-(2-benzylmorpholin-4-yl)-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
1-butyl-5-(3-methoxy-4-methylphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-4-methylpyrimidine
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[2-(methylsulfanyl)pyrimidin-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-phenoxypropanamide
(1R,5R)-N,N-dimethyl-6-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-cyclopentyl-4-{1H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
1-[2-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-cyclopentyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-{4-[(2,2-dimethyloxan-4-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
2-({[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-N-(2,4-dimethylphenyl)acetamide
1-(2-{1-[(3-chloro-1H-indol-2-yl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-(4-hydroxy-2-methylquinolin-6-yl)benzamide
N-(2-methyl-5-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)butanamide
N-[(1S,2R)-2-aminocyclobutyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
[3-(2-methoxyethyl)-1-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl]methanol
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(1-benzofuran-2-sulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
methyl 2-(benzylsulfamoyl)-6-[(3,4-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4,6-dimethyl-2-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydropyridine-3-carboxamide
1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-N-(oxan-4-ylmethyl)piperidin-4-amine
1-[2-({[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
2-(4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenoxy)pyrimidine
2-{[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}-2-methylpropan-1-ol
{1-[(3-methylquinoxalin-2-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylcyclopropane-1-carboxamide
6-(2-methoxyphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyridazin-3-amine
3-[({1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-3-yl}oxy)methyl]pyridine
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(methylsulfanyl)phenyl]methyl})amine