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2-(6-hydroxypyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-N-(diphenylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[(3S,4R)-1-(5-chloropyridin-2-yl)-4-propylpyrrolidin-3-yl]acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
3-(5-{2-[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}quinazolin-4-amine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
9-(4-cyclobutyl-6-methylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-cyclopentyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-methoxyphenyl)methyl]acetamide
N-(cyclohexylmethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-[2-(2-fluorophenyl)ethyl]piperidine
1-(3,5-dimethylfuran-2-carbonyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
5-(2-hydroxybenzoyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[5-(2-carbamoylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-[4-(benzylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-[(2-hydroxyethyl)sulfamoyl]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
{1-[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}(pyridin-2-yl)methanol
1-[4-(3-fluorophenoxy)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
N-{2-[2-(6-chloro-2-fluoro-3-methoxyphenyl)-1H-imidazol-1-yl]ethyl}acetamide
2-{[(1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-(1-methoxypropan-2-yl)-1-(2,3,5,6-tetramethylbenzoyl)piperidine-4-carboxamide
N-[(2,3-dimethylphenyl)methyl]-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-{[4-(5-propylpyrimidin-2-yl)piperazin-1-yl]methyl}benzoic acid
2-methyl-6-{[1-(3-methylphenyl)piperidin-4-yl]amino}heptan-2-ol
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-benzyl-1H,2H,3H,4H,5H-pyrido[3,2-b]indol-2-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
4-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-[2-(2,6-difluorophenyl)ethyl]-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
N-({5-[3-(methylsulfanyl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-8-methoxyquinoline
1-(dimethyl-1,3-thiazole-4-carbonyl)-4-methanesulfonyl-1,4-diazepane
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(morpholin-4-yl)propan-1-one
3-{4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]phenyl}propanoic acid
2-{2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
(4aS,8aS)-2-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-decahydroisoquinolin-4a-ol
N-(2-methoxyethyl)-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)propanamide
2-(1,4-dithiepan-6-yl)-8-methyl-2,8-diazaspiro[4.5]decane
(4-{[1-(dimethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-4-(2-methoxyphenyl)piperazine-1-carboxamide
4-benzyl-1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-(furan-3-ylmethyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-methyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-[(3-methylthiophen-2-yl)sulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
1-cyclohexanecarbonyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrrolidine-2-carboxamide