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4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(2-phenylethyl)piperidin-4-yl}methanol
4-[(2,6-dimethoxyphenyl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
5-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-N-(oxan-4-ylmethyl)piperidin-4-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H-pyrazole-3-carboxamide
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-[(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
4-[5-(2-hydroxyethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1-methyl-1,2-dihydroquinolin-2-one
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-{4-[4-(hydroxymethyl)phenyl]-1H-pyrazol-1-yl}acetamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-fluorobenzene-1-sulfonamide
2-methoxy-5-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}pyridine
(1R,3S)-3-methoxy-7-[(trimethyl-1H-imidazol-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(2-phenylethyl)piperidine
3-({2-amino-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)-N-(2-methoxyphenyl)propanamide
4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-N-methylbenzene-1-sulfonamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
(2S,4S)-4-(4-{2-[(3-fluoro-4-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(but-3-enoyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[3-(propan-2-yloxy)benzoyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
4-(5-chloro-2-ethoxyphenyl)-1-ethyl-5-methyl-1H-pyrazole
(3aS,7aR)-5-methyl-2-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
6-chloro-1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-cyclopentyl-4-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
1-[(4aS,8aS)-7-cyclohexyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-methylbut-2-en-1-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzene-1-sulfonamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
ethyl 4-benzyl-1-[(2,3-difluorophenyl)methyl]piperidine-4-carboxylate
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
1-(2-methanesulfonylethyl)-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-1-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
3-(benzenesulfonyl)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
4-(4-fluorophenyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-ol
4-ethyl-3-({1-[(3-hydroxy-6-methylpyridin-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
4-[(1E)-3-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
(3S,4S)-1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl})[2-(pyridin-4-yl)ethyl]amine
4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(2S,4R)-4-(dimethylamino)-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidine-2-carboxylic acid
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-{[(3,4,5-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
4-hydroxy-N,1-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
2-(dimethylamino)-4-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrimidine-5-carboxamide