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ethyl 4-[(4-chlorophenyl)methyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxylate
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-propylpiperidine
methyl N-(1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-1-oxopropan-2-yl)carbamate
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N,N-dimethylpyrrolidin-3-amine
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
(1S,5R)-3-(1,3-benzothiazol-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,2-dimethyloxan-4-yl)-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-(2-aminoethyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
6-{[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]amino}-N,N-dimethylpyrazine-2-carboxamide
1-[(4-fluorophenyl)methyl]-4-(4-methylpyrimidine-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-[(2-hydroxyadamantan-2-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[3-(methylsulfanyl)propyl]urea
3-{2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-(3-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}phenyl)-1H-pyrazole
(3S,4R)-1-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-[(1-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}piperidin-4-yl)methyl]benzoic acid
(1,4-dioxan-2-ylmethyl)({2-[(2-fluorophenyl)methoxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)amine
4-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-methylpyrimidine
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
2-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
(4aR,7aS)-1-(2-methylpropyl)-4-(1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3,4-dimethoxyphenyl)amino]-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-methylbutyl)piperidine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[2-(trifluoromethyl)benzoyl]piperidin-3-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
2-(3-chlorophenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide
{9-[3-(methylsulfanyl)propyl]-3-(pyridine-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-(3-propyl-1H-pyrazole-5-amido)pyrrolidine-3-carboxylic acid
1-{1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}-4-phenylbutane-1,4-dione
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
(2R,6R)-4-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
6-(2-methyl-1,3-thiazol-4-yl)-2-[4-(piperazin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-benzyl-4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1H-pyrazole
1-[(3-fluorophenyl)methyl]-4-(piperidin-3-ylmethyl)piperazine
4-(2-methoxyphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(6-methoxypyridin-2-yl)phenol
2-[2-(3-methoxyphenyl)ethyl]-4-{3-[2-(pyridin-3-yl)piperidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(4-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}piperidin-1-yl)ethan-1-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(4aS,7aR)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[3-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-dimethyl-1H-pyrazole
1-(2-methoxybenzoyl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(N-methylmethanesulfonamido)propanamide
N-(3-cyanophenyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-[(2-butoxy-3-methoxyphenyl)methyl]-1-methanesulfonylpiperidin-4-amine
5-(2-chlorophenyl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]furan-2-carboxamide