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dimethyl(2-{2-[1-(propane-2-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
5-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
6-methyl-N4-[1-(2-phenylethyl)piperidin-4-yl]pyrimidine-2,4-diamine
3-(2-phenylethyl)-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
4-[2-(4-acetylphenoxy)acetyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
3-(azepane-1-sulfonyl)-5-(1H-1,2,3-benzotriazol-1-yl)benzoic acid
N-cyclopropyl-2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]pyridine-4-carboxamide
N-[(4-methylphenyl)methyl]-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
2-[N-methyl-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]-2-(pyridin-3-yl)acetic acid
N-[2-(dimethylsulfamoyl)ethyl]-1,3-benzothiazole-6-carboxamide
(3S,4R)-1-[(2,4-difluorophenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
4-[4-(1H-indole-6-carbonyl)piperazin-1-yl]quinazoline
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-(pyridin-2-ylmethyl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]piperidin-2-one
N-(1H-indol-6-ylmethyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
ethyl 1-(prop-2-en-1-yl)-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-methyl-2-oxo-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-acetyl-N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)thiophene-3-carboxamide
2-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]pyridine-3-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-ethyl-2-(1-{[(1-methyl-1H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)benzamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(1H-indol-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2,3-dihydro-1-benzofuran-5-carboxamide
1-{5-[(benzyloxy)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}butan-2-ol
1,3-dimethyl-2,6-dioxo-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-methyl-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
2-[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-N-cyclopropylacetamide
N-[1-({methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
3-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoic acid
methyl[2-(morpholin-4-yl)propyl][(2-phenyl-1H-imidazol-4-yl)methyl]amine
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-methyl-3-phenylbutan-1-one
7-cyclopentyl-2-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(4aR,7aS)-1-methyl-4-[4-(2-oxopyrrolidin-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridin-3-ol
methyl 3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[(4,4-difluoropiperidin-1-yl)methyl]-2-(methylsulfanyl)pyrimidine
(1S,5R)-6-(2-methoxyethyl)-3-(1-phenylcyclopentanecarbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2,3,6-trimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethan-1-ol
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
[3-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)-2,2-dimethylpropyl]dimethylamine
N-({1-[(3-chloro-2-methylphenyl)carbamoyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
4-{1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
N-{1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]pyrrolidin-3-yl}-N-methylacetamide
1-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]propyl}-4-(3-chlorophenyl)piperazine