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N-[3-(2-methoxyphenyl)-3-methylpentyl]-4-methylpyrimidine-5-carboxamide
3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
(1S,5R)-6-(1-methyl-1H-pyrazole-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S)-3-{4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}azepan-2-one
3-(3,4-dimethoxybenzoyl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
3-{2-[4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-indole
(1R,5S,6S)-6-{4-[2-(4-chloro-2-methylphenoxy)ethyl]piperazine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
2-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
1-[1'-(2,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]urea
2-(3-methoxypropyl)-8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-acetamido-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)thiophene-2-carboxamide
7-chloro-3-methyl-2-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1H-indole
2-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-3-methylquinoxaline
1-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-cyclopropyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
3-{1-[1-(3-fluoropropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
3-(3,4-dichlorophenyl)-N-methylpyrazin-2-amine
4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
3-propanamido-N-[1-(thiophen-2-yl)propyl]benzamide
4-[4-(piperidine-1-carbonyl)phenoxy]-1-(thian-4-yl)piperidine
2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(3-ethylphenyl)acetic acid
1-cyclobutanecarbonyl-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]piperidine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
(3aR,6aR)-2-acetyl-5-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(2-methoxyethyl)(methyl)[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]amine
(2S,4S)-N-ethyl-4-[(naphthalen-1-ylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[3-(cyclopropylmethyl)-1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl]methanol
1-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
(4aS,7aR)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-(2,4,6-trimethoxyphenyl)-1H-imidazole
1-[3-(benzyloxy)piperidin-1-yl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2,6-dimethylphenyl acetate
N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(pyridin-2-yl)propanamide
3-({4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)benzonitrile
3-(cyclobutylmethoxy)-5-[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]benzoic acid
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(1-benzofuran-5-ylmethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-(cyclopropylmethyl)-4-(pyridine-3-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
1-cyclopentyl-N-(2-hydroxyethyl)-5-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-3-carboxamide