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1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
4-[1-(2-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
6-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
3-chloro-N-[2-(pyridin-3-yloxy)propyl]thiophene-2-carboxamide
(1R,2S)-N1-tert-butyl-N2-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]cyclohexane-1,2-dicarboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
1-cyclopropyl-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[(3-methyloxetan-3-yl)methyl]amine
6-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
5-[5-(1-benzyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[(3,4-difluorophenyl)methyl]-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
1-[(2,3-difluorophenyl)methyl]-3-({[(2,5-difluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
5-fluoro-2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
1-(2-methanesulfonylethyl)-2-(1-phenylethyl)-1H-imidazole
1-(1-benzyl-4-phenylpiperidine-4-carbonyl)azetidin-3-ol
3-({4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
3-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
2-amino-4-(3,4-dihydroxyphenyl)-6-(1-ethyl-1H-indol-3-yl)pyridine-3-carbonitrile
N-[(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrrole-2-carboxamide
N-tert-butyl-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamido]-2-methylbenzamide
4-[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]-N-(furan-2-ylmethyl)pyridine-2-carboxamide
1-(2-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}morpholin-4-yl)ethan-1-one
1-ethyl-N-[2-(3-fluorophenyl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-tert-butyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(butan-2-yl)-N3-butyl-N5-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methoxypyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-[(2-methylpyridin-3-yl)oxy]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(thiophene-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aS,7aR)-5-methyl-2-(1-methylcyclohexanecarbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(azepan-1-yl)-3-(3-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
N-methyl-2-(methylsulfanyl)-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
N-(1-{4-[2-(4-fluorophenoxy)ethyl]phenyl}ethyl)acetamide
(1r,4r)-4-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
2-[(1S,5R)-6-(3-chloro-4-hydroxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(1S,6R)-9-[2-methyl-2-(morpholin-4-yl)propyl]-3,9-diazabicyclo[4.2.1]nonane
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-hydroxy-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
2-methoxy-N-{3-[4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]phenyl}benzamide
1-methyl-2-oxo-N-(oxolan-2-ylmethyl)-6-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]pyrimidin-2-amine
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-chlorophenyl)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethan-1-ol
1-(3-methoxy-3-methylbutyl)-5,5-diphenylpiperidin-2-one
7-(3-ethyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine