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N-({1-[(3-acetylphenyl)methyl]piperidin-4-yl}methyl)-2-methylpropanamide
(3S,4S)-1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidine-3,4-diol
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
6-(2,6-dimethoxyphenyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(1H-imidazol-2-yl)-4-phenyl-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
(1R,5S,8S)-N,N-dimethyl-3-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
1-{3-[3-(quinolin-3-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(piperidin-1-yl)piperidine-1-carboxamide
1-(oxan-4-yl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-cycloheptyl-N-methyl-6-oxo-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide
6-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(3aS,6aS)-3a-(hydroxymethyl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]-octahydrocyclopenta[c]pyrrole-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-propylthiophene-3-carboxamide
N4-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]pyrimidine-4,6-diamine
N4-ethyl-N2-[1-(4-methylbenzoyl)piperidin-4-yl]pyrimidine-2,4-diamine
5-chloro-3-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-methyl-6-[2-(thiophen-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
3-ethyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-indole-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4,4-difluoro-N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-(1-methyl-1H-indazol-5-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-4-ylmethyl)urea
N-(butan-2-yl)-3,5-dimethyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-4-carboxamide
3-(pyrimidin-5-yl)quinoline
4-[4-(carbamoylmethoxy)phenyl]-N,N-dimethylbenzamide
8-(1H-imidazol-2-ylmethyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-({2-[1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
3-(3-methylphenyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]piperidine-1-carboxamide
3-[(3R,4S)-1-(2,5-dimethylfuran-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(3-chloro-4-methylbenzenesulfonyl)-4-[(dimethylamino)methyl]azepan-4-ol
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({2-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]phenyl}methyl)propanamide
1-ethyl-5-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(2-oxo-2-{3-[(6-oxo-1,6-dihydropyridin-3-yl)methyl]pyrrolidin-1-yl}ethyl)-1λ6-thiane-1,1-dione
5-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
7-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(2S)-1-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
4-[4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]but-3-yn-1-ol
2-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-3-methylbutan-1-ol
(1S,5R)-6-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-1-[(6-methylquinolin-8-yl)sulfonyl]-4-propylpyrrolidin-3-amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(1R,5R)-6-(cyclopropylmethyl)-3-(4-methoxy-3-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane