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1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
[1-(cyclohex-1-ene-1-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
3-(4-hydroxyphenyl)-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4,4-difluoropiperidine
1-[2-(1H-imidazol-5-yl)ethyl]-3-[(2-methoxyphenyl)methyl]-5-(oxolan-3-yl)-1H-1,2,4-triazole
4,4-difluoro-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidine
1-{4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenyl}ethan-1-ol
N-[4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenyl]acetamide
2-(2-ethoxypyridin-3-yl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
ethyl 2-{methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}acetate
3-chloro-4-{[1-(cyclobutylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-(4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-(3-phenylpropyl)piperazin-2-yl)ethan-1-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(2-methoxyphenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-pyrazole-4-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
7-[cyclohexyl(methoxy)methyl]-4-(thiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(2-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
N-cycloheptyl-1-cyclopropyl-5-[4-(2-methylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[2-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)phenyl]-1λ6-thiomorpholine-1,1-dione
6-{3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
N-({1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}methyl)acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(morpholin-4-yl)pyrimidine-5-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
1-[6-(pyrimidin-5-yl)-1,2,3,4-tetrahydroquinolin-1-yl]ethan-1-one
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
(3aS,6aS)-2-methyl-5-[(6-methylquinolin-8-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
7-(cyclopropylmethyl)-2-(4-methylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(benzylsulfamoyl)-5-bromobenzoic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3R,4R)-4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-3-ol
(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-({[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)amino)propane-1,2-diol
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-3-ylmethyl)pyridin-2-amine
[(3R,4R)-1-(5-fluoro-2-methoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(2R,3R,6R)-5-(furan-2-carbonyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(4-chlorophenyl)ethyl]-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[3-(4-hydroxyphenyl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{3-oxo-3-[4-(2-phenoxyethyl)piperazin-1-yl]propyl}azepan-2-one
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N,2-dimethyl-2-{methyl[(2-phenylphenyl)methyl]amino}propanamide
[(3R,4R)-1-(3-chloro-2-fluorobenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(4,6-dimethylpyridin-2-yl)-3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylphenol
(2,1,3-benzoxadiazol-5-ylmethyl)[(2-cyclohexylpyrimidin-5-yl)methyl]methylamine
9-(2H-1,3-benzodioxol-5-ylmethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(oxolan-2-ylmethyl)amine