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methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperazine
(3S,4R)-4-(2-methoxyphenyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(3-fluorophenyl)methyl]-1,4-diazepane
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(thiomorpholin-4-yl)propan-1-one
N-[2-(2,4-difluorophenyl)-1-[1-(thiophene-3-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
5-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)-6-methyl-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
5-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
3-[4-(4-fluorophenyl)-4-oxobutyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
4-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]-1-(3-methoxyphenyl)piperazin-2-one
3,5-dimethyl-4-[5-({3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
(1S,5R)-6-(4-fluoro-2-methylbenzenesulfonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(quinolin-3-ylmethyl)(thiophen-2-ylmethyl)amino]butan-1-ol
N-[(3S,5S)-1-acetyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-chloro-1H-indole-2-carboxamide
4-methoxy-N-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]benzene-1-sulfonamide
N5-cyclopropyl-N6-(prop-2-en-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
5-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4-phenylpyrimidin-2-amine
N-ethyl-6-(3-fluoro-4-methoxyphenyl)pyridazin-3-amine
(1S,5R)-6-benzyl-3-[5-(hydroxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2-phenoxyethyl)piperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-[(4-chlorophenyl)(phenyl)methyl]-6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{3-[3-(2,5-dimethylfuran-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}ethan-1-one
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
4-{[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-2-yl]methyl}morpholine
1-tert-butyl-4-[4-(2,4-difluorophenyl)-5-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
2-(2-chloro-4-fluorophenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-{[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]pyrrolidine-3-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}ethan-1-one
(2E)-3-(1,3-benzothiazol-2-yl)-1-[3-(5-methyl-1,2-oxazol-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]prop-2-en-1-one
N-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1-ethylpyrrolidin-3-amine
4-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-(1-methylazepane-2-carbonyl)piperidine-4-carboxylate
ethyl 4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}-1H-pyrazole-3-carboxylate
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
7-(furan-3-ylmethyl)-N4-[2-(1H-pyrrol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethyl-2-(1H-pyrrol-1-yl)propanamide
2-chloro-6-fluoro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}benzamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3,5-dimethylbenzoyl)piperidine
2-[4-(pyridin-3-yloxy)piperidin-1-yl]-2-(thiophen-3-yl)acetic acid
N-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]methyl}-2-hydroxy-2-methylpropanamide
ethyl 2-(3-acetamidophenyl)pyridine-3-carboxylate
4-ethyl-5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-(furan-2-yl)-5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}pyrimidine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroquinolin-2-one
(1R,2R,6S,7S)-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane