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1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2-{1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]piperidin-2-yl}ethyl)dimethylamine
methyl 6-(2-cyclopropylacetyl)-2-{[(4-methylphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methoxy-N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(3S,4R)-4-(hydroxymethyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-ol
2-(4-methylphenyl)-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
methyl 1-{3-[(cyclopropylmethyl)amino]-5-(pyrrolidine-1-sulfonyl)benzoyl}piperidine-2-carboxylate
4-[(2S,3R)-2-amino-3-hydroxybutanoyl]-1-(2-phenylphenyl)piperazin-2-one
3-{3-[({[(2-methoxy-5-methylphenyl)carbamoyl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(3S,4R)-1-[3-(dimethylamino)benzoyl]-4-methylpiperidine-3,4-diol
2-(methylamino)-1-[4-(thiomorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidine
2-{4-[(ethylcarbamoyl)methyl]piperazin-1-yl}-N-(propan-2-yl)pyridine-4-carboxamide
3-methyl-3-phenyl-1-[4-(thian-4-yl)piperazin-1-yl]butan-1-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-methoxy-4-(prop-2-en-1-yl)piperidine
3-(3-methylthiophen-2-yl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]propanoic acid
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4,5-dimethyl-2-(1H-1,2,3,4-tetrazol-1-yl)thiophene-3-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
(2S,4S)-N-[(4-methylphenyl)methyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-4-(1H-pyrazol-3-yl)benzamide
2-(2,6-difluoro-4-methoxyphenyl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
5-(1-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-2-yl)thiophene-2-carboxylic acid
7-[(1E)-pent-1-en-1-yl]-1,2-dihydroisoquinolin-1-one
3-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)quinoline
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-ol
1-methyl-5-({2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3,4-tetrazole
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2-{4-[1-(3-chloro-2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)urea
8-[(4-chloro-3-fluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-[4-(2-hydroxyethyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(3R,4S)-4-{4-[6-(piperidin-1-yl)pyrimidin-4-yl]-1,4-diazepan-1-yl}oxolan-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(2-methoxyethoxy)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
3-methyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
2-[4-(2-amino-5-ethylpyrimidin-4-yl)-1-(furan-3-ylmethyl)piperazin-2-yl]ethan-1-ol
7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(4-fluorophenyl)-1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperidin-4-ol
2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}-N-[2-(1H-pyrazol-4-yl)ethyl]pyridine-3-carboxamide
3-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
3-[(methylsulfanyl)methyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
7-(cyclobutylmethyl)-2-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
4-[(4-fluorophenyl)methyl]-1-[(4-methoxypyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(2R,3R,6R)-3-(4-methylphenyl)-5-(trimethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-4-amino-N-ethyl-1-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}urea