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3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(3-phenylpropanamido)phenyl]propanamide
2-methyl-7-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
ethyl 1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyridin-4-yl)ethyl]amine
1-(dimethylamino)-3-(4-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperazin-1-yl)propan-2-ol
4-hydroxy-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-(6-methyl-2H-1,3-benzodioxol-5-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-methyl-3-phenyl-N-(thian-4-yl)-1H-pyrazole-4-carboxamide
3-(3-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}phenyl)-N,N-dimethylpropanamide
6-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]-2,3,4,5-tetrahydropyridazin-3-one
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methoxy-6-methylbenzamide
N-(3-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}phenyl)acetamide
1-(2-chlorophenyl)-3-{1-[1-(2-hydroxybutyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
[(3R,4R)-1-(2-amino-9H-purin-6-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-(benzyloxy)-8-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1,8-diazaspiro[4.5]decan-2-one
(3aR,6aR)-2-(3,5-dimethoxybenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-tert-butyl-2-({3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}methyl)phenol
8-{[3-(furan-2-yl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-methyl-1-(3-oxo-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propyl)-1,2-dihydropyridin-2-one
1-ethyl-6-oxo-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
(3R,4S)-1-(8-chloroquinolin-2-yl)-4-propylpyrrolidin-3-amine
2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)pyridine-3-carboxamide
7-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-yl]methanol
N-ethyl-2-{4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}acetamide
5,6-dimethoxy-2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-methyl-3-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(4-fluorophenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}phenyl)pyridine
3-[(cycloheptylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine
2-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-8-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(2R,3R)-1'-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
5-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-1H-1,2,3-benzotriazole
1-[1-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
N-[(2-chlorophenyl)methyl]-3-[1-(pyrimidin-5-ylmethyl)piperidin-3-yl]propanamide
4-{2-oxo-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-1-yl}benzonitrile
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-phenyl-2-(piperidin-1-yl)ethyl]butanamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-(pyrrolidin-1-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
N-({5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2,5-dimethyl-3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-(3,5-dimethylphenyl)-4-(pyridin-3-ylmethyl)piperazin-2-one