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1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[1-(2-methylpropyl)cyclopropyl]amino}methyl)piperidin-2-one
1-[({5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}amino)methyl]cyclohexan-1-ol
4-{[3-(carbamoylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[2-(3,4-difluorophenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
2-(4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)-1,3-benzothiazole
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-oxazole-3-carboxamide
N-(4-{4-[ethyl(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
1-{3-[1-(2-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-methoxy-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(1R,3S)-3-ethoxy-7-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-[4-(3-methylphenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
1-{[4-(pyridin-2-yl)phenyl]methyl}-4-(pyridin-3-yl)piperazine
N-cyclohexyl-2-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}butanamide
1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
(3S,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(4-chlorophenoxy)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
5-methyl-2-(4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}piperidin-4-yl)pyridine
1-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-3-phenylpropan-1-ol
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
1-(2-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,4-dihydropyridin-4-one
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-[1-methyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-3-yl]pyridine
5-(azepane-1-carbonyl)-N-methyl-1-(2-methylpropyl)-4-oxo-N-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(azepan-1-yl)-3-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)propan-2-ol
1-{1-[6-(4-fluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]ethan-1-one
5-(methanesulfonylmethyl)-2-(2-methoxy-5-methylphenyl)pyridine
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-methyl-1-(3-{[(6-methylhept-5-en-2-yl)amino]methyl}piperidin-1-yl)propan-1-one
4-({1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}methyl)morpholine
N-(1-{[(2,2-diphenylethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
5-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2,4-triazin-3-amine
3-[5-(2-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-[(3-chlorophenyl)methyl]-4-[4-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
7-(cyclobutylmethyl)-2-(1-methylpiperidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-butyl-4-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperazin-2-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,4-dioxan-2-ylmethyl)-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
N-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(3,4-dichlorophenyl)-4-[6-(morpholin-4-yl)pyrimidin-4-yl]morpholine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-2-(3-methyl-1H-pyrazol-5-yl)pyridine
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-3-(2-oxoazepan-1-yl)propanamide
N-ethyl-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(4-chlorobenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(1-benzyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(1-methyl-1H-pyrazole-4-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine