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7-(cyclopropylmethyl)-N-(2-hydroxypropyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1S,5R)-3-(3-phenylpropyl)-6-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(2,4-diethoxy-3-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(4aR,7aS)-1-benzyl-4-(furan-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-methoxyphenoxy)-1-(1H-pyrrole-3-carbonyl)piperidine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
4-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-3-yl}benzoic acid
1-(azepan-1-yl)-3-[3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
6-methyl-N-{1-oxaspiro[4.5]decan-3-yl}imidazo[1,2-a]pyridine-2-carboxamide
1-methyl-2-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-(4-{[4-(quinoline-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
N-(2-chloro-3,5-difluorophenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-8-methoxyquinoline
4-phenyl-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
4-(2,3-dihydro-1H-inden-2-yl)-11-{[(2-fluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
8-(4-methanesulfonylphenyl)quinolin-4-amine
2-(1-ethyl-1H-indazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[1-(4-pentyl-1H-1,2,3-triazol-1-yl)ethyl]-1,3,4-thiadiazol-2-amine
6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydropyridazin-3-one
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-(dimethylamino)-8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-(3-chlorophenyl)-N-[2-(pyrazin-2-yl)ethyl]-1,2,4-triazin-3-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[2-(3-phenylpiperidin-1-yl)ethyl]urea
3-(1-methylpiperidin-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
3-[5-(ethanesulfonyl)thiophen-2-yl]-2-methoxypyridine
6-(benzyloxy)-1-(2-methylpropyl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one
N-[(5-methylpyrazin-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
[3-(4-methyl-1H-pyrazol-1-yl)propyl](4-phenylbutan-2-yl)amine
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(2-methoxyphenyl)benzoyl]pyrrolidin-3-yl]methanol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-cyclopropyl-1H-pyrazole-5-carboxamide
7-fluoro-4-[2-(3-methoxypropyl)piperidine-1-carbonyl]-2-methylquinoline
1-[5-(2-methoxybenzoyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
3-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]azetidin-3-yl}pyridine
3-cycloheptyl-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(thiophen-2-yl)-1,2,4-oxadiazole
2-[4-(cyclopropylmethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
dimethyl({5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amine
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(2-methoxyethoxy)ethan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
1-(1'-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[1-(dimethylamino)cyclopentyl]methyl}acetamide
1-(4-phenylpiperazine-1-carbonyl)-6-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane
2-(4-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-(5-acetyl-2-ethoxyphenyl)-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide