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[2-(furan-2-yl)ethyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
(3S,4S)-1-(1,3-benzothiazole-6-carbonyl)-4-[benzyl(methyl)amino]pyrrolidin-3-ol
2-[(2H-1,3-benzodioxol-4-ylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(4-methyl-2-oxo-2H-chromen-7-yl)-2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carboxamide
3-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-hydroxy-3-methylbutyl)-N-[2-(1-hydroxycyclopentyl)ethyl]benzamide
2-[4-(propan-2-yl)morpholin-2-yl]-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)acetamide
4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-2-methoxyphenol
2-(4-ethylpiperazin-1-yl)-N-[2-(3-methylpyridin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(dimethyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[6-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)pyrimidin-4-yl]piperidin-4-ol
1-[5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-ethyl-7-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.4]nonane
N-ethyl-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-(1-hydroxybutan-2-yl)-N-(thiophen-2-ylmethyl)-2-(thiophene-2-sulfonamido)acetamide
2-{1-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]-1H-imidazol-2-yl}benzoic acid
3-cyclopropyl-5-(4,5-dimethylthiophen-2-yl)-1-ethyl-1H-1,2,4-triazole
2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
N-[(3-methylphenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aR,7aS)-1-(2-methylpropanoyl)-4-(5-methylpyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
4-[(2,3-dimethoxyphenyl)methyl]piperazine-2-carboxylic acid
(1S,5R)-3-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]imidazo[1,2-a]pyridine-2-carboxamide
(4aR,7aS)-1-ethyl-4-[6-(hydroxymethyl)pyridine-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(4-methoxy-3-methylphenyl)pyrazin-2-amine
({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-(2-chloro-3-methoxyphenyl)-3-[2-(pyrrolidin-1-yl)ethyl]urea
({4-ethyl-5-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-{4-[2-(ethylamino)ethoxy]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
N-(3-hydroxy-3-phenylpropyl)-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-(2-methylpropyl)-3-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
3-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
methyl 4-(3-hydroxyphenyl)-1-methyl-1H-pyrrole-2-carboxylate
1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
N-cyclopropyl-3-methoxy-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
1-(1H-imidazol-4-ylmethyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-(3-hydroxy-3-phenylpropyl)-N,5-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[1-(6-methylpyridin-3-yl)ethyl]pyridin-2-amine
3-(5-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-6-(methoxymethyl)pyridine-2-carboxamide
N-[2-(1H-pyrazol-1-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]oxane-4-carbonitrile
9-[3-(benzyloxy)propyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one