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3-{[2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]methyl}benzoic acid
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methylpentanamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{5-cyclopentyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(furan-2-carbonyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,4-diazepane
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-3-(piperidin-3-yl)benzamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
ethyl 1-{[3-(furan-3-amido)-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-3-carboxylate
(3S,4R)-3-ethyl-4-methyl-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperidin-4-ol
2-butoxy-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-2-(1H-imidazol-2-yl)-N-methylbenzamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
4-{5-[3-(2-methylphenyl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
1-(3-fluorophenyl)-3-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[(5-chloro-2-hydroxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
8-[3-(1-methyl-1H-pyrrol-2-yl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-{4-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
5-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-N-(propan-2-yl)pyrimidin-2-amine
1-[5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]propan-1-one
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(1,3-thiazol-2-yl)benzamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-hydroxyethyl)piperidine-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
4-[(5-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-propylpiperidine
3-[(2R,5R)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazine-1-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
1-(morpholin-4-yl)-3-[5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-ethyl-2-methyl-1,3-thiazole-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(4-methylphenyl)propanamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]cyclopropanecarboxamide
N-[1-(3,4-difluorophenyl)piperidin-4-yl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[(4-fluorophenyl)methyl]-4-(2-methyl-1,3-thiazole-4-carbonyl)morpholine
N-cyclopropyl-1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(3R,4R)-4-ethyl-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidine-3,4-diol
3-(dimethylamino)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
methyl 2-(3-{3-[3-(dimethylcarbamoyl)phenyl]phenyl}-1H-pyrazol-1-yl)acetate
6-methyl-2-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(thiophen-3-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-({2-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1,4-dimethyl 2-[2-(2,4-dimethylbenzenesulfonamido)acetamido]butanedioate
2-(2-methoxyethoxy)-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol