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2-(2-aminoacetyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(4-methanesulfonylphenyl)-1,2,3,4-tetrahydroisoquinoline
6-[(1-methylpiperidin-4-yl)amino]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-ethoxyphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-{[(thiophen-2-ylmethyl)carbamoyl]methyl}pyrrolidine-3-carboxylic acid
1-{2-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]phenyl}ethan-1-one
3-(2-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
4-cyclobutyl-6-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
2-(4-fluorophenyl)-4-[4-(1H-imidazol-1-yl)benzoyl]morpholine
(isoquinolin-5-ylmethyl)({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-(2-methylpropyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-1-[1'-(pyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-cyclopropyl-2-[3-(4-methylphenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
5-cyclopropanecarbonyl-1'-(2-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoacetamide
2-{4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
S-(4-fluoro-3-methylphenyl)-2-(3-methoxypiperidin-1-yl)-2-oxoethane-1-sulfonamido
N-[2-(ethylsulfanyl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
5-(4-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
5-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
[(3,4-dimethoxyphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-methyl-6-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1H-indole
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
1-methyl-N-[2-(propylsulfanyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
(3aR,6aS)-N-[2-(3-phenylpropoxy)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
4-(3,4-diethoxyphenyl)-2-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
4-({4-methyl-5-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
5-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[(4-fluorophenyl)methyl]-N-[2-(1H-indol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(5S,9aS,9bS)-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(5-chloropyridin-2-yl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)piperazine-1-carboxamide
8-[(3-chloro-4-fluorophenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
6-(4-ethyl-5-methylthiophene-3-carbonyl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
6-{[methyl(2-phenylethyl)amino]methyl}-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
{5-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
2-[5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-(3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1-benzofuran-2-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amine
3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-[2-(dimethylamino)ethyl]-6-methyl-2-(2-phenylethyl)-1,4-dihydropyridin-4-one
N-benzyl-2-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3-methylthiophen-2-yl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine