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1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
4-(4-fluoro-2-methylphenyl)-1-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-1,2,3-triazole
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-[(4-methoxyphenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]acetamide
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(3-fluoropyridin-4-yl)-7-azaspiro[3.5]nonan-1-ol
3-{5-[1-(3-methoxybenzoyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
3-amino-1-({4-[2-oxo-2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyrrolidine-3-carboxylic acid
7-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-(2-chloropyridin-3-yl)-3-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]urea
6-(2-chlorophenyl)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2,5-trimethylfuran-3-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
3-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,5-dimethyl-1H-pyrazole
3-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-4-(pyrrolidine-1-carbonyl)piperidine
2-[4-(4-methylpiperazin-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(thiophen-2-yl)propan-2-yl]acetamide
6-[4-(pyrrolidin-1-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N,N-diethyl-2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-sulfonamide
2-chloro-3-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-6-methoxyphenol
3-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanoic acid
1-(4-chlorophenyl)-4-(3-hydroxypyridine-2-carbonyl)-5-methylpiperazin-2-one
benzyl(cyclopropylmethyl){[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
(1R,9S)-11-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-oxo-N-[4-(pyridin-2-yl)butyl]-1,2-dihydroquinoline-4-carboxamide
5-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(2S)-2-[4-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]-3-methylbutanamide
methyl 6-benzoyl-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-5-[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
N-[(2,4-dimethoxyphenyl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(2R,3R,6R)-5-(2,4-dimethylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-benzoyl-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3aR,6aR)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(2-fluorophenyl)methyl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazin-2-one
4-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(pyridin-3-yl)morpholine
N-[3-(2-methoxyacetamido)-2-methylphenyl]-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2E)-4-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-2-enamide
4-benzyl-3-ethyl-1-(4-hydroxy-3-methoxybenzoyl)-1,4-diazepan-5-one
3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-(oxan-4-yl)benzamide
2-[(4-chlorophenyl)methyl]-N-(2-hydroxybutyl)-1,3-benzoxazole-5-carboxamide
3-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
3-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1-methylimidazolidine-2,4-dione
N-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
3-benzyl-1-(1,3-thiazol-2-yl)piperidine-3-carboxylic acid