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[(3aS,6aS)-2-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
3-butanamido-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}benzamide
(1R,3S)-7-[(3,4,5-trimethoxyphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
1-[(2-methylnaphthalen-1-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
3-(2-methylphenyl)-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
4-hydroxy-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
3-[(dimethylamino)methyl]-1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-3-ol
7-(cyclopropylmethyl)-2-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-{[1-(6-methylpyridin-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S,4R)-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-(3-aminopropanoyl)-5-butyl-1-(3-phenylphenyl)piperazin-2-one
N-(1-methyl-1H-indazol-5-yl)-4-(pyridin-4-yl)piperidine-1-carboxamide
4-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperazin-2-one
(2S,4R)-4-(2,2-dimethylpropanamido)-N,N-diethyl-1-(1H-pyrrole-3-carbonyl)pyrrolidine-2-carboxamide
1-(2-phenylethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
1-(cyclohexylmethyl)-N,N-dimethyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(morpholine-4-sulfonyl)-5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]benzoic acid
(3aR,5R,6S,7aS)-2-{[4-(2-fluorophenyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}piperidine-4-carboxamide
(1-{1-[(6-methoxynaphthalen-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
N-(1-benzyl-1H-pyrazol-3-yl)-2-(4-methyl-1H-pyrazol-1-yl)acetamide
(2R)-2-{5-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propanamide
ethyl 4-({4-[(2H-1,3-benzodioxol-5-yl)amino]-8-methylquinazolin-2-yl}methyl)piperazine-1-carboxylate
5-{4-[(2-ethylmorpholin-4-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-(furan-2-yl)pyrimidine
(3R,4R)-4-(azepan-1-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-ol
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(3R)-piperidin-3-yl]-1H-1,3-benzodiazole-5-carboxamide
1'-(3-fluoropyridin-4-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2-methoxyethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,3-dihydro-1H-inden-1-yl)-1,2-oxazole-3-carboxamide
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-(4-methylpentan-2-yl)piperidine
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
5,7-dimethyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N,1-dimethyl-3-(2-methylpropyl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
N-[(3R,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(oxane-4-carbonyl)pyrrolidine-2-carboxamide
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1'-(5,6-dimethylpyrimidin-4-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[5-(1-carbamoylcyclopropyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-ethylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(6-phenoxypyridin-3-yl)-1-(pyridin-2-ylmethyl)piperidine-2-carboxamide
1-[(4-methoxyphenyl)methyl]-5-[(2R)-oxolane-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N,N-dimethyl-4-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperazine-1-sulfonamide
N-cyclopentyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(2-methylphenyl)methyl]propanamide
7-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one