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9-[2-(1-methylpiperidin-2-yl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
7-methyl-4-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-(4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-1-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(3aS,6aS)-2-[2-(2-chloro-6-fluorophenyl)acetyl]-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(2-phenylethyl)piperidine
5-(2-chloro-5-methylbenzoyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2,5-dimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-2-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}pyrimidin-4-amine
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[2-(propan-2-yl)phenyl]urea
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
4-[(4-hydroxypiperidin-1-yl)methyl]-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)benzamide
4-(2-fluoro-5-methylphenoxy)-1-(morpholine-2-carbonyl)piperidine-4-carboxylic acid
3-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-(3,4,5-trimethoxyphenyl)urea
2-(1H-pyrazol-1-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]butan-1-one
2-(9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
4-methyl-1-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-triazole
4-(4-fluorobenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
N-[4-methoxy-2-(2-methylpropanamido)phenyl]piperidine-3-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-[2-(methylamino)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5-(methanesulfonylmethyl)pyridine
1-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-4-(thiophen-2-yl)butan-1-one
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-(2-oxopiperidin-1-yl)propanamide
3,3-dimethyl-1-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}urea
5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
1'-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
[1-({1-[(2E)-2-methylpent-2-en-1-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-(dimethylamino)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
3-(hydroxymethyl)-1-(1-phenylcyclopentanecarbonyl)piperidin-3-ol
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}thiophene-3-sulfonamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-3-ethylpiperidin-3-ol
4-(2-fluoro-5-methylphenoxy)-1-(furan-3-ylmethyl)piperidine-4-carboxylic acid
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
[(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
2-amino-8-(6-methoxy-2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-{4-cyclopentyl-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidine-4-carbonitrile
2-(3-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-6-methoxypyrimidin-4-amine
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(2-methoxyethoxy)ethan-1-one