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2-(3,4-dimethoxyphenyl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
1-(3,5-dimethylphenyl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazin-2-one
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-methoxy-1-{4-[(2-methoxy-4-methylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}ethan-1-one
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
N-[2-(dimethylamino)ethyl]-5-(1,2,5-oxadiazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-(1-pentanoylazepan-3-yl)propanamide
1-(piperidine-1-sulfonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
1-ethyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
3-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-(2,5-difluorophenyl)-2-[2-(1-ethylpiperidin-4-yl)acetamido]acetic acid
3-{2-oxo-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}imidazolidine-2,4-dione
1-[(6-methoxypyridin-3-yl)methyl]-4-(pyridin-2-ylmethyl)piperazine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-ethyl-5-methyl-1H-pyrazole-3-carboxamide
2-{5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
1-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]thiophen-2-yl}ethan-1-one
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-3-[3-(methoxycarbonyl)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{2-propoxy-5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]phenyl}methanol
2-(2,6-dimethoxyphenyl)-N-propylbenzamide
N-(3-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
5-(4-acetyl-2-methoxyphenoxymethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
methyl[(3-methylthiophen-2-yl)methyl]{[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
[(1R,3S,3aS,6aR)-3-(2-chloro-4-fluorophenyl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-cycloheptyl-2-(1-ethyl-1H-pyrazol-4-yl)-N-methylquinoline-4-carboxamide
1-{1-[3-amino-6-(2-methylquinolin-5-yl)pyrazin-2-yl]piperidin-4-yl}-2-methylpropan-1-ol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
(3S,4S)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4,5-trimethoxyphenyl)acetamide
(3S,4S)-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-methylpiperidine-3,4-diol
3-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-(2,5-dimethylphenyl)urea
N-butyl-3-(2-hydroxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
6-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridin-6-yl]pyrazine-2-carboxamide
(1S,5R)-6-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-methyl-1,3-thiazol-2-amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(4-fluoro-3-methoxyphenyl)methyl](2-methoxyethyl)amine
3-acetamido-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
3,4,7-trimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-indole-2-carboxamide
(1R,5S,8R)-3-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
2-ethyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrimidine
3-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
9-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[3-(morpholin-4-yl)propyl]piperidine-3,5-dicarboxamide
2-butoxy-1-[6-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[3-(dimethylamino)phenyl]-4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
1-methyl-4-{2-[3-(pyridin-2-yl)azetidin-1-yl]pyridine-4-carbonyl}piperazine
(2S,4R)-4-amino-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-benzyl-8-[2-(morpholin-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one