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3-(2-{[3-(3-methoxyphenyl)phenyl]carbamoyl}piperidin-1-yl)propanoic acid
N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
(2S)-2-amino-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1,3-thiazol-4-yl)propanamide
5-[(3-methoxypyrrolidin-1-yl)methyl]-2-(pyrrolidin-1-yl)-1,3-thiazole
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(pyridin-4-yl)ethan-1-one
2-(pyridin-3-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S,4S)-1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-3,4-diol
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2-methoxyphenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4R)-3-hydroxy-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl]pyrazine-2-carboxamide
5-{[3-(2-methoxy-5-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
4-fluoro-N-({1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl}methyl)benzamide
2-(4-ethylpiperazin-1-yl)-N-[1-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-methyl-7-(1,2-oxazole-3-carbonyl)-N-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-(benzyloxy)ethan-1-one
2-[(2-amino-5-ethylpyrimidin-4-yl)amino]-N,N-dimethylethane-1-sulfonamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-phenylpropan-1-one
N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
2-methyl-4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}phenol
4-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
3-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-N-methylpyridin-2-amine
(2S)-1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methyl-2-(methylamino)pentan-1-one
7-fluoro-4-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-methylquinoline
4-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidine-1-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
3-(pyrazin-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
4-cyclopropanecarbonyl-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-[4-(3-fluorophenoxy)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
(3R,4S)-3,4-dimethyl-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-4-ol
3-[({2-[3-(trifluoromethyl)phenyl]ethyl}amino)methyl]piperidin-3-ol
6,6-dimethyl-1-(2-methylphenyl)-N-[(2,3,4-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
(2S)-3-methyl-2-[(3-methyl-4-oxo-3,4-dihydrophthalazin-1-yl)formamido]butanamide
1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
N-ethyl-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
1-(2-methoxyethyl)-N-[(6-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-benzyl-2-(2-phenylethyl)pyrrolidine-1-sulfonamide
2-methyl-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-1-benzofuran-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
2-(propan-2-yl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
N-(1H-1,3-benzodiazol-2-ylmethyl)-N,3-dimethyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]ethan-1-one
8-[(2R)-2-aminopentanoyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1H-1,3-benzodiazol-2-ylmethyl)({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea