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N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-4-yl)methyl]quinoline-4-carboxamide
7-fluoro-2-methyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}quinoline
4-(2-hydroxy-5-methoxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-3-(piperidin-1-yl)pyridine-2-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-2-(propan-2-yl)pyrimidine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-[(cyclopropylmethyl)sulfanyl]acetamide
5-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-2-methyl-3,4-dihydropyrimidin-4-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}acetamide
2-[3-(2-methoxyphenyl)phenoxy]acetamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(furan-3-ylmethyl)-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
N-[1-(1-cyclooctylpiperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-9-oxa-2-azaspiro[5.5]undecane
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(3-phenylpiperidin-1-yl)acetamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-methyl-2-(4-methylphenoxy)propan-1-one
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-5-phenyl-1H-pyrrole
1-({3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
3-methyl-1-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)butan-1-ol
5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}pyrimidine
2-(dimethylamino)-8-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[3-(3-chlorophenyl)phenyl]-N-(1H-1,2,4-triazol-5-ylmethyl)piperidin-4-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-fluoro-N-methyl-5-sulfamoylbenzamide
1-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-1,4-diazepan-5-one
N-(1,3-benzothiazol-2-ylmethyl)-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(4-methyl-1H-pyrazol-5-yl)-1-(4-methylbenzenesulfonyl)piperidine
1-(2-phenylphenyl)-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
4-(2-methylphenoxy)-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(5-fluoro-2-methoxybenzoyl)piperidine
5-acetyl-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
4-[2-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]acetamide
3-methyl-7-(3-phenylpiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}-2-methoxyphenol
2-[3-(piperidin-3-yl)benzoyl]-2-azaspiro[4.4]nonane
3-[1-(3-hydroxybenzoyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
3,7-dimethyl-11-(2-propoxybenzoyl)-3,7,11-triazaspiro[5.6]dodecane
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-[(2-methoxyphenyl)methyl]acetamide
5-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-{1-[(2,3-dimethoxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
(3S,4S)-1-{[3-(benzyloxy)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol