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2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylacetamide
2-amino-4-methyl-N-(1-propylpyrrolidin-3-yl)pyrimidine-5-carboxamide
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(2-methoxyquinolin-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-[2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
2-{4-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-(2-hydroxyphenoxy)-N-methylacetamide
2-ethyl-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
3-(2,4-dimethoxyphenyl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
2-[(1-methylpiperidin-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
5-methyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-3-phenyl-1,2-oxazole-4-carboxamide
N-cyclopropyl-2-(ethanesulfonyl)-N-[(3-ethoxyphenyl)methyl]propanamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
4-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]phenyl}-4H-1,2,4-triazole
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-methyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3S,4S)-1-[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-(4-methoxyphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-cyclopentyl-2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4S)-1-(2,6-dimethylpyridin-4-yl)-3,3,4-trimethylpiperidin-4-ol
(3S,4S)-3-hydroxy-N-(4-methyl-3-propanamidophenyl)-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
[2-(4-{1-[3-(trifluoromethyl)phenyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)ethyl]urea
(1R,3S)-3-methoxy-7-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-{3-oxo-3-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propyl}pyrrolidin-2-one
3-[2-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
methyl 2-[1-(1-cyclopentyl-6-oxopiperidin-3-yl)-N-methylformamido]acetate
{3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
N-methyl-N-[2-(pyridin-2-yl)ethyl]azepane-4-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-{2-[1-(4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-[(dimethylamino)methyl]-1-(4-phenyl-1H-imidazole-5-carbonyl)pyrrolidin-3-ol
2-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}-N-methylacetamide
4-(hydroxymethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
[(2S,6S)-4-(5-phenyl-1,2-oxazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-acetyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[3-(3-chlorobenzoyl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
11-(2,6-dimethoxypyrimidine-4-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
ethyl 4-(3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-6H,7H,8H-cyclopenta[g]quinolin-2-yl)piperazine-1-carboxylate
2-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-yl)acetic acid
4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(3-methoxyphenyl)-1-phenyl-1H-pyrazole
(1S,6R)-N-(4-fluorophenyl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-5-[1-(methylsulfanyl)propan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
ethyl 4-(cyclopropylmethyl)-1-[(2-methyl-1H-indol-3-yl)methyl]piperidine-4-carboxylate
N-(1H-indol-4-ylmethyl)-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide