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5-(2-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
[2-(1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-2-yl)ethyl]dimethylamine
2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-6-ol
(3S,4R)-4-(pyridin-4-yl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidine-3-carboxylic acid
7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,4-dithiepan-6-amine
{1-[3-(1H-pyrazol-1-yl)benzoyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
2-[3-(propan-2-yloxy)phenyl]-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
N'-(3-chloro-4-fluorophenyl)-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]butanediamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)benzamide
4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}pyridine
N-cyclopentyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1S,5R)-3-(4-aminopyrimidin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-5-methyl-2-phenyl-1H-imidazole
4-amino-2-{4-[(5-butylthiophen-2-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
N-[4-(2-fluorophenoxy)phenyl]-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxamide
ethyl 1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]-4-(2-phenylethyl)piperidine-4-carboxylate
2-methoxy-N-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
(3R)-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-ethyl-4-(methoxymethyl)-5-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-(3-ethylmorpholine-4-carbonyl)-7-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-({[3-(cyclopentyloxy)propyl]amino}methyl)-8-fluoroquinolin-4-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
2-methyl-6-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
[1-(5-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
N-cyclopentyl-1-[1-(2-ethylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
2-(5-fluoro-4-methoxypyrimidin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(pyrrolidin-1-yl)butanoyl]piperidine-4-carboxylic acid
N-methyl-2-(propan-2-yl)-N-[1-(pyridin-3-yl)propyl]pyrimidine-4-carboxamide
4-{[methyl(thian-4-yl)amino]methyl}-1H-pyrazole-3-carboxylic acid
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-ethyl-1-[(2-fluorophenyl)methanesulfonyl]piperidine-3-carboxylic acid
[1-(cyclopent-1-ene-1-carbonyl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
5-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]pyrrolidin-2-yl}-N-(2-hydroxyethyl)thiophene-2-carboxamide
3-{1-[(3,4-difluorophenyl)methyl]-1H-imidazol-2-yl}benzonitrile
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
(3S,4S)-1-[2-(2-ethylphenoxy)ethyl]-4-methylpiperidine-3,4-diol
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-(1-cycloheptylpiperidin-3-yl)-2-(methylsulfanyl)acetamide
ethyl 4-[3-({[(2-chlorophenyl)methyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
N-[2-(1H-imidazol-1-yl)ethyl]-1-benzothiophene-5-carboxamide
3-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-2,8-diazaspiro[4.5]decane
methyl 2-({1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}sulfonyl)benzoate