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2-[4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3-(1,2-oxazolidin-2-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
7-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
2-methyl-5-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]phenol
5-cyclopropanecarbonyl-1'-(oxane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]morpholin-3-yl}acetic acid
[(4aS,8aR)-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
(1S,5R)-6-(4-chloro-3-fluorobenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-(2-chloro-6-fluorobenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(2-fluoro-5-methoxyphenyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(3-methoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-tert-butyl-4-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-methyloxane-2-carbonyl)-1,4-diazepane
ethyl 4-[3-({[(3-fluorophenyl)methyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)but-3-yn-1-ol
(1S,5R)-3-(2-acetylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{3-[1-(but-2-yn-1-yl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyrimidin-4-amine
1,2-dimethyl-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1H-indol-5-ol
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)(quinolin-6-ylmethyl)amine
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(2-ethyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2E)-3-(4-chlorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-en-1-one
1-(3-{[3-(azonane-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
6-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carboxylic acid
2-fluoro-N-({4-hydroxy-1-[(2-methyl-1,3-oxazol-4-yl)methyl]azepan-4-yl}methyl)benzamide
3-[(3,4-dimethoxyphenyl)methyl]-5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
(2S)-2-amino-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentan-1-one
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(2-methyl-1H-imidazol-1-yl)propanamide
dimethyl({3-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]propyl})amine
5-oxo-1-(pyridin-3-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
2-(pyridin-3-yl)-N-(quinolin-3-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
({4-cyclopropyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-(3-fluorophenyl)-3-{1-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[(4-fluorophenyl)methyl]-3-[1-(quinolin-8-ylmethyl)piperidin-4-yl]propanamide
3-[(4-acetyl-1,4-diazepan-1-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
5-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-cyclobutyl-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
1-ethyl-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}cyclopent-1-ene-1-carboxamide
4-{6-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidin-4-yl}morpholine
ethyl 5-{[5-(methoxymethyl)furan-2-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[2-(dimethylamino)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylthiophene-2-carboxamide
(2S,4S)-4-amino-1-{3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]propanoyl}-N-methylpyrrolidine-2-carboxamide
3-(3-methylthiophene-2-carbonyl)-N-(2-phenylethyl)piperidine-1-carboxamide
5-(3,5-difluoro-4-methoxyphenyl)-2-methoxypyridine