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2-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
N-phenyl-4-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}piperidine-1-carboxamide
1-{5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl]propan-1-ol
1-methyl-3-(2-methylpropyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
N-(2-{[(1S,3R)-3-aminocyclopentyl]formamido}ethyl)pyridine-4-carboxamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-methyl-1,3-benzoxazole
[(3-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](furan-2-ylmethyl)methylamine
N4,N4-diethyl-6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine-2,4-diamine
1-{4-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
3-methoxy-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
ethyl 1-{1-[4-(3-phenylpropanamido)phenyl]piperidin-4-yl}piperidine-3-carboxylate
ethyl 1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N3-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(cyclohex-3-en-1-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methoxyethoxy)ethan-1-one
2-(dimethylamino)-1-[8-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
(3aS,6aS)-2-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1'-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
9-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{3-[(4-methoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl}morpholine
benzyl 2-[6-oxo-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-1,6-dihydropyridazin-1-yl]acetate
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(2-phenylethyl)-6-(9H-purin-6-yl)-decahydro-1,6-naphthyridin-2-one
3-(2-methoxyethyl)-1-[(4-methylpiperazin-1-yl)sulfonyl]piperidine-3-carboxylic acid
5-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)isoquinoline
2-(dimethylamino)-2-(3-methylphenyl)-1-(morpholin-4-yl)ethan-1-one
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
1-{[1-(2,5-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-cyclopropyl-1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
4-(1H-imidazol-1-yl)-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-[2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetyl]pyrrolidine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{4-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenyl}but-3-yn-1-ol
N-[(3-methylpyridin-2-yl)methyl]-5-(phenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
3-[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]benzonitrile
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-(4-phenylbutyl)urea
4-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[3-(5-methylfuran-2-yl)benzoyl]piperidine
7-(cyclopropylmethyl)-2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-{4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}quinazoline
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[2-(methoxymethyl)-1-methyl-7-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]-2-phenylacetamide
methyl 5-[(2,3-dihydro-1H-inden-2-yl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(3-methoxyphenyl)-N-methyl-N-(pyrazin-2-ylmethyl)benzamide