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2-(ethylamino)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrimidine-5-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-[4-(hydroxymethyl)piperidin-1-yl]-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]acetic acid
4-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
2-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1,3-benzoxazole
3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-indazole
N-[4-(pyridin-2-yl)butyl]-3-azaspiro[5.5]undecan-9-amine
(4aR,7aS)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
9-(5-methyl-1,2-oxazole-3-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-(3-hydroxyquinoxalin-2-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]propanamide
2-[4-(cyclopropanesulfonyl)morpholin-3-yl]-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]acetamide
3-phenoxy-1-[4-(pyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-[(2-chlorophenyl)methyl]-2-(morpholin-2-yl)-N-(propan-2-yl)acetamide
N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-indole-6-carboxamide
8-(5-ethyl-2-methylpyrimidin-4-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-5-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]pyrimidin-2-amine
2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(3-chlorophenyl)methyl]-4-{4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
[2,4,6-trimethyl-3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenyl]methanol
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-amino-4-{[(6-chloropyridin-3-yl)methyl]amino}quinazoline-6-carboxylic acid
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(4-chloro-1-ethyl-1H-pyrazol-5-yl)-1-(4-methoxyphenyl)-1H-1,2,4-triazole
(4aS,7aR)-N-(2-chlorophenyl)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
8-[2-(4-benzylmorpholin-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-cyclopropyl-N-[1-(furan-2-carbonyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
1-ethyl-4-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-1H-pyrrole-2-carbonitrile
1-(4-phenoxybutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-N-ethyl-1-(naphthalen-2-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N-{3-[4-({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,2-oxazole
4-(3-fluorophenoxy)-1-(2-methylfuran-3-carbonyl)piperidine
1-(3-chlorophenyl)-4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine
2-methoxy-5-[1-(3-methoxypropyl)-1H-imidazol-2-yl]pyrimidine
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
methyl (2S)-2-{[1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
N-(3-{[(1-ethylpyrrolidin-3-yl)methyl]sulfamoyl}phenyl)acetamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
3-methyl-4-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}-1,2,5-oxadiazole
(1R,5R)-3-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(1-ethyl-1H-pyrazol-3-yl)phenyl]pyridine
2-butyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R)-1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}pyrrolidin-3-ol
1-(3-aminobenzoyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
4-{5-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
7-(3,6-dimethylpyrazin-2-yl)-4-[(3-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol