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1-(2,3-dihydro-1H-indene-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(3,4-dimethoxyphenyl)methyl]acetamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
2-({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
2-[4-(methylsulfanyl)phenyl]-2-[4-(pyridin-3-yloxy)piperidin-1-yl]acetic acid
4-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]butanamide
5-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
4-(6-methoxypyridin-2-yl)-2-{[(naphthalen-1-ylmethyl)amino]methyl}phenol
N-(4-methoxy-2-methylphenyl)-2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)sulfamoyl]dimethylamine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
3-(3-methoxyphenoxymethyl)-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine
4-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]-1,4-oxazepan-6-ol
2-phenoxy-1-{4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-2-methyl-1,4-diazepan-5-one
N-[2-(dimethylamino)ethyl]-3-({1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}oxy)-4-methoxybenzamide
6-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-ethyl-2-methoxy-3-{[(1-propylpiperidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(cyclopropylmethyl)-8-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-1,6-dimethyl-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydropyridin-4-one
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-[(2-methyl-1-benzothiophen-3-yl)methyl]morpholine
5-hydroxy-N-[(1r,4r)-4-methoxycyclohexyl]pyridine-2-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
1-(5-{[4-(methoxymethyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-4-methyl-1,4-diazepane
1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1,3-dimethyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
11-[(2,3-dihydro-1H-inden-2-yl)amino]-4-[2-(4-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{4-[2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-3-cyanopyridin-4-yl]phenyl}acetamide
8-fluoro-4-oxo-N-(5-oxo-1-propylpyrrolidin-3-yl)-1,4-dihydroquinoline-3-carboxamide
2-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
3-[4-fluoro-3-(hydroxymethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
5-(1-benzofuran-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,2,4-triazin-3-amine
3-cyclopentyl-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
6-[3-(2-fluorophenyl)-3-phenylpropanoyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
{1-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-yl}methanol
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[3-(4-methylphenyl)phenyl]pyrrolidine-1-carboxamide
N-ethyl-N-(2-methoxyethyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
3-[(2-methoxyethyl)sulfamoyl]-5-(1H-pyrazol-1-yl)benzoic acid
(1S,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-5-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1H-pyrrole-3-carbonitrile
5-{[4-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-methylfuran-2-carboxamide
1-methanesulfonyl-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-amine
1-cyclopropyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(ethylsulfanyl)propan-1-one