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(3R,4R)-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](ethyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclohexyl-N-methylacetamide
1-[methyl({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amino]propan-2-ol
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(methylsulfanyl)propan-1-one
{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}methanol
N-cyclohexyl-N-(pyridin-3-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[3-(4-methylpiperazin-1-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
4-(1H-imidazol-1-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}butan-1-one
2-({4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
[1-(4-aminopyrimidin-2-yl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
2-{2-[(3-acetamidopyrrolidin-1-yl)methyl]phenoxy}acetic acid
4-[4-(1-methyl-1H-imidazol-5-yl)benzenesulfonyl]thiomorpholine
2-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-7-methyl-4H-chromen-4-one
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole
5-{1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-methoxypyridine
5-{[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
3-({1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,3-dihydro-1H-indol-1-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-oxoacetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(1H-indazol-3-yl)acetamide
N-methyl-2-[3-methyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
N-(benzylsulfamoyl)-N-(pyridin-2-ylmethyl)cyclohexanamine
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-ol
(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-ethyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-{2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
dimethyl({1-[3-({methyl[2-(methylsulfanyl)ethyl]amino}methyl)phenyl]ethyl})amine
3-{[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-methyl-7-(pyrazin-2-yl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
7-(cyclobutylmethyl)-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-{2-[(4-methylpyrimidin-2-yl)oxy]hex-5-en-1-yl}thiomorpholine
1-(2-aminoethyl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1H-1,2,3-triazole-4-carboxamide
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(3-methoxybenzoyl)piperidine
2-[(1S,5R)-3-[(4-chloro-3-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(3-fluoro-4-methoxybenzoyl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
(2S,4S,5R)-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]carbamoyl}-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
5-[4-(2,5-dimethylphenyl)piperazin-1-yl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-[(3,5-dimethylfuran-2-yl)methyl]-4-phenylpiperidin-4-ol
4-[1-benzyl-5-(2,3-difluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-amine
(2S,4S)-N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-methoxyacetamido)-1-methylpyrrolidine-2-carboxamide
(3R,4R)-3,4-dimethyl-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-ol
(1-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}piperidin-3-yl)methanamine
2-[1-(2-methoxyphenoxy)propan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(1-benzofuran-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
1-({4-methyl-5-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N4,5-dimethyl-N4-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidine-2,4-diamine