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(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
2-(2-ethoxypyridin-3-yl)-2-(4-phenyl-1,4-diazepan-1-yl)acetic acid
1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(thiophen-3-yl)-1H-imidazole
5-(2-methylphenyl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
(1-{1-[3-(4-chlorophenyl)phenyl]piperidin-4-yl}piperidin-4-yl)methanol
1-ethyl-5-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
8-(3,6-dimethylpyrazin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-3-(methoxymethyl)pyrrolidine
4-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(1,2-oxazol-3-ylmethyl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyridine-4-carbonyl)-1,4-diazepane
5-methyl-1-[3-(4-methylpiperazin-1-yl)propyl]-5-phenylpiperidin-2-one
5-{[(5-ethylpyridin-2-yl)methyl](methyl)carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
methyl 5-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-acetyl-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
1-[3-(azepane-1-carbonyl)phenyl]-3-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]urea
2-[2-(4-aminoazepan-1-yl)-2-oxoethyl]-4-methyl-1,2-dihydrophthalazin-1-one
N-[4-(3-methylphenyl)phenyl]-1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidine-4-carboxamide
4-ethenyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,6-difluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
(1S,5R)-6-(2-methoxy-4-methylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[3-(dimethylamino)propyl]-2-{4-[2-(furan-2-yl)-2-oxoacetyl]morpholin-3-yl}-N-methylacetamide
3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-cyclopropyl-3-[1-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)piperidin-4-yl]propanamide
1-[({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]cyclohexan-1-ol
3-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}thiophene-2-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(morpholin-2-ylmethyl)pyrimidine-5-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(5-methylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(4-benzoylpiperazin-1-yl)-2-oxoethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
9-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
(3S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2,5-dimethylphenyl)ethan-1-one
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-cyclopentylethan-1-one
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
N-(1-methyl-1H-pyrazol-5-yl)-5-[1-(4-methylpyridine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-(2-methoxy-6-methylphenyl)-3-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
5-({2-[3-(4-carboxyphenyl)piperidin-1-yl]acetamido}methyl)furan-2-carboxylic acid
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-{2-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(3,4-dichlorophenyl)morpholin-4-yl]propan-1-ol
3-{2-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one