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N,N-dimethyl-5-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
4-(2-methyl-6-propylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-methoxy-4-[(5-methylfuran-2-yl)methyl]-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-(2-methoxyethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine-4-carboxylate
5-{[benzyl(methyl)amino]methyl}-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-1-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
1-{2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-benzotriazole
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl]propylamine
[(3S,7S)-5-(5-methylpyrazine-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
2-{1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[5-(1-cyclooctylpiperidin-4-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
2-methyl-6-[3-(pyridin-3-yloxy)propyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
ethyl 1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxylate
1-[(3S,4R)-1-[2-(3-chlorophenoxy)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2-{4-[4-(propan-2-yloxy)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-4-(1H-pyrazol-1-yl)butan-2-ol
3-{4-[2-(morpholin-3-yl)acetamido]phenyl}-1H-pyrazole-5-carboxylic acid
1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-3-yl}benzoic acid
5-phenyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-ethylacetamide
7-chloro-N,3,5-trimethyl-N-[3-(morpholin-4-yl)propyl]-1-benzofuran-2-carboxamide
6-(propan-2-yl)-N-[3-(pyridin-4-yl)propyl]pyrimidin-4-amine
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(3-fluorophenoxy)ethan-1-one
ethyl 4-[4-(4-methylphenoxy)piperidine-4-carbonyl]piperazine-1-carboxylate
(4-aminobutyl)({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amine
N-butyl-N-[(2-fluorophenyl)methyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(3-methylthiophen-2-yl)methyl]piperidine
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
6-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-2-methyl-3,4-dihydropyrimidin-4-one
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
2-(2-fluoro-5-methoxyphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
(3S,4R)-3-ethyl-4-methyl-1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]piperidin-4-ol
2-(4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
2-(2-chlorophenyl)-N-(3-methoxypropyl)-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
N-cyclohexyl-2-methyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-4-carboxamide
ethyl 5-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidine-3-carboxylic acid
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-(2-aminoethyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}quinazolin-4-amine
5-{[5-(oxan-2-yl)furan-2-yl]methyl}-3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{1-[({[4-(morpholin-4-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2H-1,3-benzodioxole-5-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3,4-difluorophenyl)methyl]benzamide
3-cyclopropyl-5-(oxolan-3-yl)-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
1-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidin-4-yl}pyrrolidin-3-ol