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5-[1-(4-methoxyphenyl)cyclopropyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
ethyl 5-(1H-1,3-benzodiazol-2-ylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(1-benzofuran-2-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4-(5-methylfuran-2-yl)-1H-1,2,3-triazole
(2S,4S)-4-amino-1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
N-[2-(benzyloxy)phenyl]-3-methoxypyrrolidine-1-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)azepane-1-sulfonamide
3-[(4-fluoro-3-methoxyphenyl)methyl]-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 2-(2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
N-{[4-(3,4-dimethylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
(3R,5R)-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-[6-(3-methoxyphenoxy)pyridin-3-yl]-1-[2-(morpholin-4-yl)ethyl]urea
1-(2-methylphenyl)-2-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)propanamide
2-[2-(pyridin-4-yl)ethyl]-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(5-methyl-1H-pyrazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-(2-chlorobenzamido)-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
3-{[(cyclopropylmethyl)(2-methoxyethyl)carbamoyl]amino}-2-methylbenzamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(2-oxopiperidin-1-yl)acetamide
methyl 4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-(oxolan-3-yl)-5-(4-phenyl-1,3-thiazol-2-yl)-1,2,4-oxadiazole
3-(azepane-1-carbonyl)-N,N-diethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[(4-fluorophenyl)methyl](methyl)amino}-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
3,3-diphenyl-1-(pyrrolidine-3-carbonyl)piperidine
2-oxo-8-[3-(pyrazin-2-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(4-methylphenyl)methyl]-4-{2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetyl}piperazin-2-one
2-(4-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}phenyl)ethan-1-amine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(4-methoxypyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
1-[(3,5-dichloropyridin-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(thiophen-2-yl)acetamide
2-{5-[5-(hydroxymethyl)furan-2-yl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}acetic acid
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(2-methylpyridine-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
3-(furan-2-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
4-ethoxy-N-[(6-methylpyridin-2-yl)methyl]benzamide
6-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]quinoline
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
1-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
N-[(1R)-1-(4-methoxyphenyl)ethyl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-phenyl-1-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethan-1-ol
1-{1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethan-1-ol