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N-[2-(benzyloxy)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-{1-[2-(4-fluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
methyl 1-(cyclopropylmethyl)-2-oxo-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
5-(3-acetylphenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-(1H-imidazol-2-yl)-N-{2-[methyl(2-phenylethyl)amino]ethyl}benzamide
2-{4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-1-yl}-1,3-benzothiazole
(2E)-3-(4-methoxyphenyl)-1-[4-(3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
(2-chlorophenyl)methyl 2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(2,5-dimethoxyphenyl)methyl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-2-methyl-N-(oxan-4-ylmethyl)-6-(piperidin-3-yl)pyrimidin-4-amine
4-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
2-(4-acetyl-1,4-diazepan-1-yl)-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]acetic acid
5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridin-2-amine
(3R,5S)-N3-(4-fluorophenyl)-N5-[(3-fluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
ethyl 4-[2-(2-phenylethyl)-1,3-benzoxazole-5-carbonyl]piperazine-1-carboxylate
1-(methoxymethyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}cyclobutane-1-carboxamide
1-[2-methoxy-5-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-{4-[({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)sulfamoyl]phenyl}acetamide
2-(2-methoxyethyl)-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(furan-2-ylmethyl)acetamide
methyl 3-(2-chlorobenzamido)-5-{[(2,2-dimethyloxan-4-yl)formamido]methyl}benzoate
1-(ethanesulfonyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
5-(cyclopropylmethyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclobutanecarbonylpiperidin-3-ol
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)benzoic acid
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]ethan-1-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
(2S,4S)-4-amino-N-methyl-1-[2-(4-methylbenzoyl)benzoyl]pyrrolidine-2-carboxamide
1-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
[1-(1,3-dimethyl-1H-indole-2-carbonyl)-3-propylpiperidin-3-yl]methanol
8-[(2,3-dimethoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[(2-cyanophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{9-[2-(3-fluorophenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
methyl 6-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyrimidine-4-carboxylate
1-{1-[2-(2-chloro-4-fluorophenyl)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-9-(1-phenylcyclopentanecarbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
6-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
4-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
N-(4-{1-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
2-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N-(prop-2-en-1-yl)pyridine-3-carboxamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-3-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
1-(2,3-dimethylphenyl)-N-[(3-methylquinoxalin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1'-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one