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5-cyclobutanecarbonyl-1'-(pyridin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(2-methylphenyl)-4-[(2-methylpyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(3,3-diphenylpiperidin-1-yl)-1-oxopropan-2-yl]methanesulfonamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2-(pyridin-4-ylsulfanyl)acetamide
1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
methyl 4-(4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)benzoate
3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
(3S,9aR)-3-(4-aminobutyl)-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-9H-purin-6-amine
N-cyclopropyl-4-methoxy-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzamide
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
N,N-dimethyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-fluorophenyl)-5-[(2-methoxy-4-methylphenyl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-hydroxy-3-methylbutan-1-one
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}propanamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-5-methyl-1-propyl-1H-pyrazole
3-{2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]ethyl}-2,3-dihydro-1H-indol-2-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(1-methyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
(1S,6R)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]sulfamoyl})amine
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
methyl 6-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}pyridine-3-carboxylate
2-{1-[(4-fluorophenyl)methyl]-4-[(2E)-2-methylbut-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-(thiolan-3-yl)piperidin-4-amine
5-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-N-methylpyrimidin-2-amine
N-(4-fluorophenyl)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
N-ethyl-N-(2-hydroxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
4-benzyl-3-ethyl-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1,4-diazepan-5-one
1-[2-(trifluoromethyl)morpholin-4-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
6-cyclopentyl-N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentanecarboxamide
3-phenoxy-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
2-{2-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1H-pyrrol-1-yl}pyridine
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
8-[(2-carboxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
5-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-3-ol
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,7aR)-1-(1-methyl-1H-indole-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(4-methoxyphenyl)ethyl]-4-{[(5-methylfuran-2-yl)methyl]amino}pyrrolidin-2-one
1-{1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxo-N-phenylacetamide
2-ethoxy-5-(2-{[(6-methylpyridin-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid