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2-(1H-1,3-benzodiazol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)acetamide
2-methoxy-4-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyridine-3-carbonitrile
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-4-(1H-pyrazol-4-yl)butanamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(1-methoxypropan-2-yl)propanamide
N-[(2-methoxyphenyl)methyl]-6-(2-methylpropyl)-2-oxo-N-propyl-1,2-dihydropyrimidine-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-methoxy-N-{2-oxo-4-[4-(prop-2-en-1-yloxy)phenyl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-propanoylpiperidine-3-carboxamide
2-[(1E)-pent-1-en-1-yl]-3-(pyrrolidine-1-carbonyl)pyridine
1-[2-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpyrrolidine-1-carbonyl)quinoline
1-cyclopentyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-(prop-2-en-1-yl)-2-[(prop-2-en-1-yl)amino]-N-(pyridin-2-ylmethyl)benzamide
1-[(3-{[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
8-[3-(dimethylamino)benzoyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(2S)-2,3-dihydro-1H-indole-2-carbonyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]urea
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]acetamide
2-(piperidin-4-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}acetamide
3-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-{4-[4-(2-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
5-(3-chlorophenyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-triazin-3-amine
6-methyl-2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridin-3-ol
1-[(6-chloropyridin-3-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide
2-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-indole
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-ol
(4aR,7aS)-1-(3-methylbutanoyl)-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
3-methyl-7-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-3,4-dihydroquinazolin-4-one
(1-{2-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
N-methyl-2-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
1-(2-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(butane-1-sulfonyl)-4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine
N-(2,3-dimethylphenyl)-2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]acetamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(phenylamino)pyrimidine-5-carboxamide
6-[4-(3,4-dichlorophenyl)piperazin-1-yl]pyrimidin-4-amine
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
ethyl 3-benzyl-1-[2-(methoxycarbonyl)benzenesulfonyl]piperidine-3-carboxylate
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(1,2-oxazol-3-ylmethyl)amine
2-{4-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
2-methyl-9-(2-methylpyrimidine-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-1-methyl-5-(2-phenoxyacetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(cyclopentyloxy)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-(3-cyclohexylpyrrolidine-1-carbonyl)-1-(2-phenylethyl)-1H-1,2,3-triazole