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2-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-5-ethylpyridine
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-4-(piperidin-1-yl)butanamide
6-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]pyridine-2-carboxylic acid
N,N-dimethyl-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-sulfonamide
4-benzyl-3-[1-(2-hydroxypyridine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidin-4-yl}pyrrolidin-2-one
2-acetyl-8-(benzenesulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4-methyl-1,2-dihydroquinolin-2-one
(4aS,7aR)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
benzyl(butyl){[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-N-{[4-(trifluoromethoxy)phenyl]methyl}propanamide
(3S,4R)-4-(hydroxymethyl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-ol
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(pyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methoxy-N,4-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
5-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(2-methylpropyl)piperidin-2-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-fluoro-2-(2-fluoro-3-methylphenyl)-4-(pyrrolidin-1-yl)pyrimidine
2-(4-fluoro-2-methylphenyl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]acetamide
4-methyl-6-(4-{[(4-phenyloxan-4-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
5-fluoro-N,N-dimethyl-2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidin-4-amine
4-[1-(2,3-difluoro-6-methoxybenzoyl)piperidin-3-yl]benzoic acid
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[4-(propan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
N2,N4,N4,5-tetramethyl-N2-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidine-2,4-diamine
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}acetic acid
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-2-amine
2-{5-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
4-(3-amino-1H-1,2,4-triazole-5-amido)-N-ethylpiperidine-1-carboxamide
1-[(6-methylpyridin-2-yl)methyl]-6-[(3-methylquinoxalin-2-yl)methyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(4-chlorophenyl)-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]morpholine
N-[(1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}piperidin-4-yl)methyl]acetamide
N-methyl-4-(pyridin-2-yl)-N-(quinolin-2-ylmethyl)pyrimidin-2-amine
1-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-3-ol
6-ethyl-1,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(4S)-4-(methoxymethyl)-1-[3-(3-methoxyphenyl)benzoyl]-3,3-dimethylpiperidin-4-ol
5-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(dimethyl-1,2-oxazol-4-yl)urea
9-[(2-ethylphenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
(1R,3S)-3-(2-aminoethoxy)-7-(1,7-dimethyl-1H-indole-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-4-oxobutane-1-sulfonamide
7-(1-benzothiophen-3-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1λ6-thiane-1,1-dione
N-benzyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-sulfonamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethan-1-one
4-(2-chloro-6-fluoro-3-methylbenzoyl)-1-(4-methoxyphenyl)piperazin-2-one
6-[(3S)-3-hydroxypyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide