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methyl (1R,3S,3aR,6aS)-3-(3-chloro-5-fluoro-4-methoxyphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-(2,5-dimethoxyphenyl)-1-(7-methyl-1-benzofuran-2-carbonyl)pyrrolidine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(propane-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{2-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-1,2,4-triazole
6-(2-aminoethyl)-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethylpyrimidin-4-amine
N-(2,2-dimethylpropyl)-N-ethyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-methyl-1H-indole-6-carboxamide
5,6-dimethyl-2-(2-oxo-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
N-[2-(piperidin-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]furan-3-carboxamide
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
{[(1R,5S,6R)-3-(furan-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-yl]methanol
1-(5-fluoropyridin-3-yl)-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
(4aR,7aS)-1-acetyl-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-3-amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-(3-ethoxy-2-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(4,4,4-trifluorobutanoyl)piperidine-2-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-phenylbenzoyl)pyrrolidin-3-yl]methanol
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[4-(oxan-2-ylmethoxy)phenyl]urea
8-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(pyrimidin-4-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{[5-(2,3-dichlorophenyl)furan-2-yl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol
2,5-dimethyl-N-{[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}furan-3-carboxamide
1-(3,5-difluorophenyl)-N-(1-propylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-(propan-2-yloxy)-N4-[1-(pyrazin-2-yl)propan-2-yl]pyrimidine-2,4-diamine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-ethylpyridine
1-(1,2-oxazol-3-ylmethyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-methyl-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
5-[3-(piperidin-1-yl)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(methylsulfanyl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-[(8-chloroquinolin-2-yl)methyl]-3-ethylpiperazin-2-one
2-oxo-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
N-(butan-2-yl)-2-(methylamino)-N-(pyridin-4-ylmethyl)benzamide
2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
1'-(propan-2-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
3-(3-fluorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
3-[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]propan-1-ol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-phenyl-1,2-oxazole-5-carboxamide
N-(oxolan-3-ylmethyl)-2-(pyridin-3-yloxy)aniline
N-cyclopentyl-4-methoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
N-ethyl-2-[(1E)-pent-1-en-1-yl]benzamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-methyl-3-phenylbutanamide
1-{[(1-methyl-1H-pyrazol-3-yl)carbamoyl]methyl}-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
7-(2-methylphenyl)-4-(piperidin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[2-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]-3-methyl-2-oxopiperazin-1-yl}acetic acid